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Diseases
Inhibitor-Anchor Map
Family Anchors
Kinase-Inhibitor Family
Template
Protein
Surface
Ribbon
Inhibitor
ATP Location
Pocket
ATP
NLP
HAP
CLP
SP
6 GSK3B related diseases
hsa05160
Hepatitis C
hsa05162
Measles
hsa05164
Influenza A
hsa05169
Epstein-Barr virus infection
hsa05215
Prostate cancer
hsa05217
Basal cell carcinoma
Summary of query kinase
Query kinase
GSK3B (
P49841
)
Kinase group
CMGC
Number of conformation types
2
Number of structural templates
24 (
Total 1039 inhibitors
)
Number of GSK3B related diseases
6 (
hsa05160
hsa05162
hsa05164
hsa05169
hsa05215
hsa05217
)
Select
Template
Comformation
Type
No. of
Templates
Representative
Template
Kinase
Group
Representative
Inhibitor
Inhibitor
Type
No. of
Kinases
No. of
Inhibitors
No. of
Diseases
A
23
1Q3DA_STU
(GSK3B)
CMGC
staurosporine
I
115
71
61
A
1Q3DA_STU
(GSK3B)
CMGC
staurosporine
I
115
71
61
115
71
61
A
2OW3A_BIM
(GSK3B)
CMGC
LY_333531
I
62
139
51
62
139
51
A
1UV5A_BRW
(GSK3B)
CMGC
6-bromoindir...
I
27
37
28
27
37
28
A
1Q3WA_ATU
(GSK3B)
CMGC
alsterpaullone
I
24
28
19
24
28
19
A
3I4BA_Z48
(GSK3B)
CMGC
Z48
I
18
77
34
18
77
34
A
1R0EA_DFN
(GSK3B)
CMGC
HMS3401D14
I
17
17
17
17
17
17
A
1PYXA_ANP
(GSK3B)
CMGC
Phosphoamino...
I
16
7
33
16
7
33
A
1J1CA_ADP
(GSK3B)
CMGC
Adenosine-5'...
I
16
7
33
16
7
33
A
1J1BA_ANP
(GSK3B)
CMGC
Phosphoamino...
I
16
7
33
16
7
33
A
3SD0A_TSK
(GSK3B)
CMGC
3-(5-Fluoro-...
I
9
38
17
9
38
17
A
1Q41A_IXM
(GSK3B)
CMGC
INDIRUBIN-3'...
I
9
25
10
9
25
10
A
3L1SA_Z92
(GSK3B)
CMGC
AN-988/42110...
I
5
33
9
5
33
9
A
3F88A_3HT
(GSK3B)
CMGC
SMR000144908
I
4
3
9
4
3
9
A
3Q3BA_55E
(GSK3B)
CMGC
ZINC13780154
I
3
3
13
3
3
13
A
1Q4LA_679
(GSK3B)
CMGC
I-5
I
3
26
7
3
26
7
A
1Q5KA_TMU
(GSK3B)
CMGC
AR-A014418
I
2
4
6
2
4
6
A
3M1SA_DW1
(GSK3B)
CMGC
HB12
I
2
3
7
2
3
7
A
3GB2A_G3B
(GSK3B)
CMGC
SB_203580
I
2
16
6
2
16
6
A
3DU8A_553
(GSK3B)
CMGC
Pyrrolopyrid...
I
2
3
6
2
3
6
A
2JLDA_AG1
(GSK3B)
CMGC
AG1
I
2
3
6
2
3
6
A
1O9UA_ADZ
(GSK3B)
CMGC
9-Methyladen...
I
1
1
6
1
1
6
A
3F7ZA_34O
(GSK3B)
CMGC
34O
I
1
15
6
1
15
6
A
3PUPA_OS1
(GSK3B)
CMGC
OS1
I
1
1
6
1
1
6
B
1
2O5KA_HBM
(GSK3B)
CMGC
2o5k
I
1
8
6
B
2O5KA_HBM
(GSK3B)
CMGC
2o5k
I
1
8
6
1
8
6