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Diseases
Inhibitor-Anchor Map
Family Anchors
Kinase-Inhibitor Family
Template
Protein
Surface
Ribbon
Inhibitor
VX3
ATP Location
Pocket
ATP
NLP
HAP
CLP
SP
Selected template
Kinase
PIM1 (PDB code: 3BGZ)
[PDB]
[PDBsum]
Inhibitor
2,3-diphenyl-1H-indole-7-carboxylic acid (HET code: VX3)
[PDB]
Summary of KIF 3BGZA_VX3
(PIM1, PDB code:
3BGZ
, chain A)
Number of family interactions
25
Number of family kinase
9 (
sequence conservation
) (
profiling results
)
Number of family inhibitors
14 (7 are PIM1 inhibitors)
Involved diseases
8 (
show
)
Number of family anchors
All kinase-inhibitor interactions in this family
PIM1 and 7 inhibitors