Protein Surface  Ribbon
Inhibitor M77
  ATP Location
Pocket ATP NLP HAP CLP SP
Selected template
Kinase ROCK1 (PDB code: 2ESM) [PDB] [PDBsum]
Inhibitor HMS2231N23 (HET code: M77) [PDB]
 
Summary of KIF 2ESMA_M77 (ROCK1, PDB code: 2ESM, chain A)
Number of family interactions 21
Number of family kinase 6 (sequence conservation) (profiling results)
Number of family inhibitors 15 (6 are ROCK1 inhibitors)
Involved diseases 24 (show)
Number of family anchors  
All kinase-inhibitor interactions in this family  ROCK1 and 6 inhibitors