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KIDFamMap
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Diseases
Inhibitor-Anchor Map
Family Anchors
Kinase-Inhibitor Family
Template
Protein
Surface
Ribbon
Inhibitor
R78
ATP Location
Pocket
ATP
NLP
HAP
CLP
SP
Selected template
Kinase
PLK1 (PDB code: 2RKU)
[PDB]
[PDBsum]
Inhibitor
BI 2536 (HET code: R78)
[PDB]
Summary of KIF 2RKUA_R78
(PLK1, PDB code:
2RKU
, chain A)
Number of family interactions
103
Number of family kinase
37 (
sequence conservation
) (
profiling results
)
Number of family inhibitors
59 (11 are PLK1 inhibitors)
Involved diseases
35 (
show
)
Number of family anchors
All kinase-inhibitor interactions in this family
PLK1 and 11 inhibitors