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KIDFamMap
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Example1
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Diseases
Inhibitor-Anchor Map
Family Anchors
Kinase-Inhibitor Family
Template
Protein
Surface
Ribbon
Inhibitor
ATP Location
Pocket
ATP
NLP
HAP
CLP
SP
Summary of query kinase
Query kinase
EPHA3 (
P29320
)
Kinase group
TK
Number of conformation types
2
Number of structural templates
6 (
Total 83 inhibitors
)
Select
Template
Comformation
Type
No. of
Templates
Representative
Template
Kinase
Group
Representative
Inhibitor
Inhibitor
Type
No. of
Kinases
No. of
Inhibitors
No. of
Diseases
B
5
2QO7A_ANP
(EPHA3)
TK
Phosphoamino...
I
18
13
59
B
2QO7A_ANP
(EPHA3)
TK
Phosphoamino...
I
18
13
59
18
13
59
B
2QO9A_ANP
(EPHA3)
TK
Phosphoamino...
I
18
13
59
18
13
59
B
2QOCA_ANP
(EPHA3)
TK
Phosphoamino...
I
18
13
59
18
13
59
B
2QOQA_ANP
(EPHA3)
TK
Phosphoamino...
I
18
13
59
18
13
59
B
3FXXA_ANP
(EPHA3)
TK
Phosphoamino...
I
18
13
59
18
13
59
E
1
3DZQA_IFC
(EPHA3)
TK
Nilotinib
II
9
30
22
E
3DZQA_IFC
(EPHA3)
TK
Nilotinib
II
9
30
22
9
30
22