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Diseases
Inhibitor-Anchor Map
Family Anchors
Kinase-Inhibitor Family
Template
Protein
Surface
Ribbon
Inhibitor
ATP Location
Pocket
ATP
NLP
HAP
CLP
SP
14 MAPK10 related diseases
H00606
Early infantile epileptic encephalopathy
hsa04930
Type II diabetes mellitus
hsa05120
Epithelial cell signaling in Helicobacter pylori infection
hsa05131
Shigellosis
hsa05132
Salmonella infection
hsa05133
Pertussis
hsa05142
Chagas disease (American trypanosomiasis)
hsa05145
Toxoplasmosis
hsa05152
Tuberculosis
hsa05160
Hepatitis C
hsa05164
Influenza A
hsa05168
Herpes simplex infection
hsa05169
Epstein-Barr virus infection
606369
Epileptic encephalopathy, Lennox-Gastaut type
Summary of query kinase
Query kinase
MAPK10 (
P53779
)
Kinase group
CMGC
Number of conformation types
2
Number of structural templates
29 (
Total 637 inhibitors
)
Number of MAPK10 related diseases
14 (
H00606
hsa04930
hsa05120
hsa05131
hsa05132
hsa05133
hsa05142
hsa05145
...
)
Select
Template
Comformation
Type
No. of
Templates
Representative
Template
Kinase
Group
Representative
Inhibitor
Inhibitor
Type
No. of
Kinases
No. of
Inhibitors
No. of
Diseases
A
3
2O0UA_C0M
(MAPK10)
CMGC
ZINC00799686
I
21
8
23
A
2O0UA_C0M
(MAPK10)
CMGC
ZINC00799686
I
21
8
23
21
8
23
A
1PMVA_537
(MAPK10)
CMGC
1,9-Pyrazolo...
I
10
5
23
10
5
23
A
3CGFA_JNF
(MAPK10)
CMGC
3cgf
I
5
15
19
5
15
19
B
26
1JNKA_ANP
(MAPK10)
CMGC
Phosphoamino...
I
15
5
27
B
1JNKA_ANP
(MAPK10)
CMGC
Phosphoamino...
I
15
5
27
15
5
27
B
1PMQA_ANP
(MAPK10)
CMGC
Phosphoamino...
I
15
5
27
15
5
27
B
3CGOA_JNO
(MAPK10)
CMGC
DB08026
I
13
32
21
13
32
21
B
1PMQA_880
(MAPK10)
CMGC
1pmq
I
12
105
20
12
105
20
B
1PMNA_984
(MAPK10)
CMGC
1pmn
I
10
124
20
10
124
20
B
2O2UA_738
(MAPK10)
CMGC
2-[(2-chloro...
I
9
19
21
9
19
21
B
2B1PA_AIZ
(MAPK10)
CMGC
AIZ
I
7
43
17
7
43
17
B
2P33A_J07
(MAPK10)
CMGC
2p33
I
6
29
19
6
29
19
B
3DA6A_BZ9
(MAPK10)
CMGC
BZ9
I
5
26
17
5
26
17
B
3PTGA_932
(MAPK10)
CMGC
N-[4-Methyl-...
I
5
19
15
5
19
15
B
3KVXA_FMY
(MAPK10)
CMGC
FMY
I
4
32
14
4
32
14
B
3OXIA_SYY
(MAPK10)
CMGC
ZINC00082427
I
4
33
16
4
33
16
B
3FI3A_JK2
(MAPK10)
CMGC
2,4-Bisanili...
I
4
6
17
4
6
17
B
3G9LX_J67
(MAPK10)
CMGC
DB08010
I
4
29
16
4
29
16
B
1PMUA_9HP
(MAPK10)
CMGC
9HP
I
4
10
17
4
10
17
B
3G9NA_J88
(MAPK10)
CMGC
DB08015
I
4
31
16
4
31
16
B
2OK1A_33A
(MAPK10)
CMGC
2oji
I
4
39
21
4
39
21
B
3OY1A_589
(MAPK10)
CMGC
5-[2-(Cycloh...
I
4
25
16
4
25
16
B
2R9SA_255
(MAPK10)
CMGC
DB06933
I
4
31
17
4
31
17
B
3G90X_J72
(MAPK10)
CMGC
CAS740841_15_0
I
4
33
16
4
33
16
B
3FI2A_JK1
(MAPK10)
CMGC
2,6-Disubsti...
I
3
4
20
3
4
20
B
2EXCX_JNK
(MAPK10)
CMGC
JNK
I
3
15
16
3
15
16
B
3FV8A_JK3
(MAPK10)
CMGC
piperazine a...
I
3
40
16
3
40
16
B
2WAJA_SNB
(MAPK10)
CMGC
CAS925681_41_0
I
1
1
14
1
1
14
B
2ZDUA_446
(MAPK10)
CMGC
EKB_569
I
1
1
14
1
1
14
B
2ZDTA_46C
(MAPK10)
CMGC
AC1NWV2E
I
1
1
14
1
1
14