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Diseases
Inhibitor-Anchor Map
Family Anchors
Kinase-Inhibitor Family
Template
Protein
Surface
Ribbon
Inhibitor
ATP Location
Pocket
ATP
NLP
HAP
CLP
SP
Summary of query kinase
Query kinase
NLK (
Q9UBE8
)
Kinase group
CMGC
Number of conformation types
0
Number of structural templates
38 (
Total 48 inhibitors
)
Select
Template
Comformation
Type
No. of
Templates
Representative
Template
Kinase
Group
Representative
Inhibitor
Inhibitor
Type
No. of
Kinases
No. of
Inhibitors
No. of
Diseases
A
34
1BL6A_SB6
(MAPK14)
CMGC
sb216995
I
46
110
50
A
1BL6A_SB6
(MAPK14)
CMGC
sb216995
I
46
110
50
46
110
50
A
1XJDA_STU
(PRKCQ)
CMGC
staurosporine
I
121
101
106
121
101
106
A
1AQ1A_STU
(CDK2)
CMGC
staurosporine
I
195
76
118
195
76
118
A
2HY81_1ST
(PAK1)
CMGC
UCN 02
I
58
20
75
58
20
75
A
1NVQA_UCN
(CHEK1)
CMGC
UCN 02
I
179
65
79
179
65
79
A
3CKXA_STU
(STK24)
CMGC
staurosporine
I
176
104
141
176
104
141
A
1NVRA_STU
(CHEK1)
CMGC
staurosporine
I
179
71
79
179
71
79
A
1NXKA_STU
(MAPKAPK2)
CMGC
staurosporine
I
110
67
51
110
67
51
A
1PKDA_UCN
(CDK2)
CMGC
UCN 02
I
195
67
118
195
67
118
A
1Q3DA_STU
(GSK3B)
CMGC
staurosporine
I
115
71
61
115
71
61
A
2C0IA_L1G
(HCK)
CMGC
A-420983
I
61
269
86
61
269
86
A
3OBGA_SB2
(MAPK14)
CMGC
SB 203580
I
21
31
28
21
31
28
A
2C0TA_L3G
(HCK)
CMGC
A-641359
I
48
260
84
48
260
84
A
1A9UA_SB2
(MAPK14)
CMGC
SB 203580
I
21
31
28
21
31
28
A
1PMEA_SB2
(MAPK1)
CMGC
SB 203580
I
16
31
26
16
31
26
A
3FMKA_FMK
(MAPK14)
CMGC
FMK
I
10
25
29
10
25
29
A
3FLNC_3FN
(MAPK14)
CMGC
Kinome_3762
I
9
44
22
9
44
22
A
3FLQA_891
(MAPK14)
CMGC
FLS
I
8
25
20
8
25
20
A
3FLSA_FLS
(MAPK14)
CMGC
FLS
I
8
26
20
8
26
20
A
3FLWA_FLW
(MAPK14)
CMGC
Pamapimod
I
9
44
22
9
44
22
A
1OUKA_084
(MAPK14)
CMGC
1ouk
I
24
139
46
24
139
46
A
3FLYA_FLY
(MAPK14)
CMGC
HMS3401N11
I
10
44
29
10
44
29
A
3FLZA_FLZ
(MAPK14)
CMGC
HMS3401P11
I
10
31
23
10
31
23
A
3FMHA_533
(MAPK14)
CMGC
FMK
I
10
25
29
10
25
29
A
1ZZLA_TZY
(MAPK14)
CMGC
CP-808844
I
36
84
44
36
84
44
A
2J90A_IZA
(DAPK3)
CMGC
Pyridone 6
I
40
50
42
40
50
42
A
2BHEA_BRY
(CDK2)
CMGC
BRY
I
51
31
35
51
31
35
A
1BL7A_SB4
(MAPK14)
CMGC
SB220025
I
22
159
29
22
159
29
A
1BMKA_SB5
(MAPK14)
CMGC
SB-218655
I
14
116
34
14
116
34
A
1OZ1A_FPH
(MAPK14)
CMGC
4-Azaindole 6
I
18
27
28
18
27
28
A
2IW6A_QQ2
(CDK2)
CMGC
2iw6
I
112
209
86
112
209
86
A
3FKOA_FKO
(MAPK14)
CMGC
L-779450
I
17
7
27
17
7
27
A
3HVCA_GG5
(MAPK14)
CMGC
HMS3303H10
I
5
76
18
5
76
18
A
2WU6A_DKI
(CLK3)
CMGC
5-AMINO-3-{[...
I
26
9
26
26
9
26
B
4
1WVYA_STU
(DAPK1)
CMGC
staurosporine
I
83
23
55
B
1WVYA_STU
(DAPK1)
CMGC
staurosporine
I
83
23
55
83
23
55
B
1H00A_FAP
(CDK2)
CMGC
AC1NAE4F
I
50
94
75
50
94
75
B
1H07A_MFP
(CDK2)
CMGC
AC1NAKJQ
I
90
241
80
90
241
80
B
1PMQA_880
(MAPK10)
CMGC
1pmq
I
12
105
20
12
105
20