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Diseases
Inhibitor-Anchor Map
Family Anchors
Kinase-Inhibitor Family
Template
Protein
Surface
Ribbon
Inhibitor
ATP Location
Pocket
ATP
NLP
HAP
CLP
SP
9 MAP2K1 related diseases
H00523
Noonan syndrome and related disorders
hsa05020
Prion diseases
hsa05034
Alcoholism
hsa05164
Influenza A
hsa05215
Prostate cancer
hsa05218
Melanoma
hsa05220
Chronic myeloid leukemia
hsa05221
Acute myeloid leukemia
115150
Cardiofaciocutaneous syndrome
Summary of query kinase
Query kinase
MAP2K1 (
Q02750
)
Kinase group
STE
Number of conformation types
1
Number of structural templates
29 (
Total 353 inhibitors
)
Number of MAP2K1 related diseases
9 (
H00523
hsa05020
hsa05034
hsa05164
hsa05215
hsa05218
hsa05220
hsa05221
...
)
Number of allelic variants
3 (
F53S
G128V
Y130C
)
Select
Template
Comformation
Type
No. of
Templates
Representative
Template
Kinase
Group
Representative
Inhibitor
Inhibitor
Type
No. of
Kinases
No. of
Inhibitors
No. of
Diseases
A
29
3EQFA_KSA
(MAP2K1)
STE
k-252a
I
42
51
57
A
3EQFA_KSA
(MAP2K1)
STE
k-252a
I
42
51
57
42
51
57
A
3EQGA_ADP
(MAP2K1)
STE
Adenosine-5'...
I
12
7
36
12
7
36
A
3EQHA_ADP
(MAP2K1)
STE
Adenosine-5'...
III
12
7
36
12
7
36
A
3EQBA_ATP
(MAP2K1)
STE
Adenosine-5'...
I
12
6
36
12
6
36
A
3EQIA_ADP
(MAP2K1)
STE
Adenosine-5'...
I
12
7
36
12
7
36
A
3E8NA_ATP
(MAP2K1)
STE
Adenosine-5'...
I
12
6
36
12
6
36
A
3DY7A_ATP
(MAP2K1)
STE
Adenosine-5'...
III
12
6
36
12
6
36
A
3MBLA_ADP
(MAP2K1)
STE
Adenosine-5'...
I
12
7
36
12
7
36
A
3ORNA_ANP
(MAP2K1)
STE
Phosphoamino...
I
12
6
36
12
6
36
A
3DV3A_ATP
(MAP2K1)
STE
Adenosine-5'...
III
12
6
36
12
6
36
A
3OS3A_ATP
(MAP2K1)
STE
Adenosine-5'...
I
12
6
36
12
6
36
A
2P55A_ATP
(MAP2K1)
STE
Adenosine-5'...
III
12
6
36
12
6
36
A
3PP1A_ATP
(MAP2K1)
STE
Adenosine-5'...
I
12
6
36
12
6
36
A
1S9JA_ATP
(MAP2K1)
STE
Adenosine-5'...
III
12
6
36
12
6
36
A
3EQDA_AGS
(MAP2K1)
STE
adenosine te...
I
11
5
27
11
5
27
A
3EQCA_AGS
(MAP2K1)
STE
adenosine te...
I
11
5
27
11
5
27
A
1S9JA_BBM
(MAP2K1)
STE
PD 0325901
III
2
28
8
2
28
8
A
2P55A_MRA
(MAP2K1)
STE
PD 0325901
III
2
12
8
2
12
8
A
3DV3A_MEK
(MAP2K1)
STE
PD 0325901
III
2
16
8
2
16
8
A
3ORNA_3OR
(MAP2K1)
STE
AKOS005266648
I
2
9
8
2
9
8
A
3MBLA_LSG
(MAP2K1)
STE
LSG
I
2
36
8
2
36
8
A
3EQHA_5BM
(MAP2K1)
STE
U0126
III
2
9
8
2
9
8
A
3EQCA_3BM
(MAP2K1)
STE
PD 0325901
I
2
25
8
2
25
8
A
3EQGA_4BM
(MAP2K1)
STE
PD 0325901
I
2
24
8
2
24
8
A
3PP1A_IZG
(MAP2K1)
STE
TAK-733
I
2
26
8
2
26
8
A
3DY7A_1CX
(MAP2K1)
STE
PD 0325901
III
1
2
8
1
2
8
A
3E8NA_VRA
(MAP2K1)
STE
PD 0325901
I
1
2
8
1
2
8
A
3EQBA_LUG
(MAP2K1)
STE
CAS881001_19_0
I
1
1
8
1
1
8
A
3OS3A_3OS
(MAP2K1)
STE
AKOS005266648
I
1
3
8
1
3
8