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Diseases
Inhibitor-Anchor Map
Family Anchors
Kinase-Inhibitor Family
Template
Protein
Surface
Ribbon
Inhibitor
ATP Location
Pocket
ATP
NLP
HAP
CLP
SP
Summary of query kinase
Query kinase
TNK1 (
Q13470
)
Kinase group
TK
Number of conformation types
0
Number of structural templates
57 (
Total 52 inhibitors
)
Select
Template
Comformation
Type
No. of
Templates
Representative
Template
Kinase
Group
Representative
Inhibitor
Inhibitor
Type
No. of
Kinases
No. of
Inhibitors
No. of
Diseases
A
35
1SM2A_STU
(ITK)
TK
staurosporine
I
99
104
128
A
1SM2A_STU
(ITK)
TK
staurosporine
I
99
104
128
99
104
128
A
1SNUA_STU
(ITK)
TK
staurosporine
I
99
104
128
99
104
128
A
1U59A_STU
(ZAP70)
TK
staurosporine
I
96
80
114
96
80
114
A
3A4OX_STU
(LYN)
TK
staurosporine
I
73
70
88
73
70
88
A
1XBCA_STU
(SYK)
TK
staurosporine
I
71
72
105
71
72
105
A
3CKXA_STU
(STK24)
TK
staurosporine
I
176
104
141
176
104
141
A
1YVJA_4ST
(JAK3)
TK
staurosporine
I
96
90
126
96
90
126
A
1BYGA_STU
(CSK)
TK
staurosporine
I
85
72
123
85
72
123
A
2DQ7X_STU
(FYN)
TK
staurosporine
I
91
74
124
91
74
124
A
1QPDA_STU
(LCK)
TK
staurosporine
I
115
76
126
115
76
126
A
2HZ4A_4ST
(ABL1)
TK
staurosporine
I
159
103
156
159
103
156
A
1QPJA_STU
(LCK)
TK
staurosporine
I
115
76
126
115
76
126
A
2XIKA_J60
(STK25)
TK
SU11652
I
59
49
65
59
49
65
A
2F4JA_VX6
(ABL1)
TK
VX-680
I
110
109
134
110
109
134
A
2XYNA_VX6
(ABL2)
TK
VX-680
I
79
101
105
79
101
105
A
3E5AA_VX6
(AURKA)
TK
VX-680
I
57
107
93
57
107
93
A
1M17A_AQ4
(EGFR)
TK
Erlotinib
I
43
166
82
43
166
82
A
2X81A_ZZL
(AURKA)
TK
MLN8054
I
22
24
64
22
24
64
A
3PJ3A_04L
(BTK)
TK
Imatinib
II
99
113
134
99
113
134
A
2C0IA_L1G
(HCK)
TK
A-420983
I
61
269
86
61
269
86
A
3EQRA_T74
(TNK2)
TK
T74
I
34
181
86
34
181
86
A
1OPLA_P16
(ABL1)
TK
PD166326
I
89
70
123
89
70
123
A
2C0OA_L2G
(HCK)
TK
A-770041
I
41
222
65
41
222
65
A
3FC2A_IBI
(PLK1)
TK
BI 2536
I
38
72
42
38
72
42
A
2FO0A_P16
(ABL1)
TK
PD166326
I
89
70
123
89
70
123
A
2C0TA_L3G
(HCK)
TK
A-641359
I
48
260
84
48
260
84
A
3KB7A_071
(PLK1)
TK
MLN_518
I
39
176
54
39
176
54
A
2G2HA_P16
(ABL1)
TK
PD166326
I
89
70
123
89
70
123
A
2HZIA_JIN
(ABL1)
TK
PD180970
I
90
77
120
90
77
120
A
1AGWA_SU2
(FGFR1)
TK
SU 4984
I
77
81
111
77
81
111
A
3FQSA_585
(SYK)
TK
R-406
I
64
28
102
64
28
102
A
2RKUA_R78
(PLK1)
TK
BI 2536
I
37
59
35
37
59
35
A
3IKAA_0UN
(EGFR)
TK
2jkk
I
76
120
108
76
120
108
A
2V7AA_627
(ABL1)
TK
5-Amido-pyrr...
I
11
23
41
11
23
41
A
3PIYA_585
(BTK)
TK
R-406
I
93
17
123
93
17
123
B
19
2ITUA_STU
(EGFR)
TK
staurosporine
I
80
85
106
B
2ITUA_STU
(EGFR)
TK
staurosporine
I
80
85
106
80
85
106
B
2ITWA_STU
(EGFR)
TK
staurosporine
I
80
85
106
80
85
106
B
3D7TA_STU
(CSK)
TK
staurosporine
I
70
68
99
70
68
99
B
3LCSA_STU
(ALK)
TK
staurosporine
I
73
100
109
73
100
109
B
2ITQA_STU
(EGFR)
TK
staurosporine
I
80
85
106
80
85
106
B
3MIYA_B49
(ITK)
TK
Sunitinib
I
70
74
110
70
74
110
B
3H10A_97B
(AURKA)
TK
MLN8054
I
39
88
82
39
88
82
B
3FUPA_MI1
(JAK2)
TK
CP690550
I
16
27
32
16
27
32
B
3EFWA_AK8
(AURKA)
TK
3efw
I
100
59
105
100
59
105
B
2WTWA_ZZL
(AURKA)
TK
MLN8054
I
35
24
70
35
24
70
B
2WKMA_PFY
(MET)
TK
PHA-665752
I
38
34
98
38
34
98
B
3EYGA_MI1
(JAK1)
TK
CP690550
I
8
23
31
8
23
31
B
3EKNA_GS3
(INSR)
TK
pyrrolo[2,3-...
I
90
215
127
90
215
127
B
2XB7A_GUI
(ALK)
TK
NVP-TAE684
I
71
66
107
71
66
107
B
2X9FA_X9F
(EPHB4)
TK
X9F
I
46
19
86
46
19
86
B
2C6EA_HPM
(AURKA)
TK
HPM
I
44
237
90
44
237
90
B
2J50A_627
(AURKA)
TK
5-Amido-pyrr...
I
11
19
34
11
19
34
B
2BMCA_MPY
(AURKA)
TK
PHA-680632
I
107
108
107
107
108
107
B
3EKKA_GS2
(INSR)
TK
pyrrolo[2,3-...
I
33
131
65
33
131
65
E
3
3G0EA_B49
(KIT)
TK
Sunitinib
I
37
40
78
E
3G0EA_B49
(KIT)
TK
Sunitinib
I
37
40
78
37
40
78
E
3G0FA_B49
(KIT)
TK
Sunitinib
I
37
40
78
37
40
78
E
2OG8A_1N8
(LCK)
TK
1N8
II
35
190
69
35
190
69