BioXGEM.
KIDFamMap
Home
Example1
Example2
Statistics
Document
Contact US
Diseases
Inhibitor-Anchor Map
Family Anchors
Kinase-Inhibitor Family
Template
Protein
Surface
Ribbon
Inhibitor
ATP Location
Pocket
ATP
NLP
HAP
CLP
SP
2 KDR related diseases
602089
{Hemangioma, capillary infantile, susceptibility to}
602089
Hemangioma, capillary infantile, somatic
Summary of query kinase
Query kinase
KDR (
P35968
)
Kinase group
TK
Number of conformation types
4
Number of structural templates
22 (
Total 2781 inhibitors
)
Number of KDR related diseases
2 (
602089
602089
)
Number of allelic variants
2 (
C482R
P1147S
)
Select
Template
Comformation
Type
No. of
Templates
Representative
Template
Kinase
Group
Representative
Inhibitor
Inhibitor
Type
No. of
Kinases
No. of
Inhibitors
No. of
Diseases
A
2
3B8RA_887
(KDR)
TK
3b8r
II
4
32
7
A
3B8RA_887
(KDR)
TK
3b8r
II
4
32
7
4
32
7
A
2P2HA_994
(KDR)
TK
triazine 34
I
3
44
19
3
44
19
B
4
3CJFA_SAV
(KDR)
TK
GW_2580
I
11
50
35
B
3CJFA_SAV
(KDR)
TK
GW_2580
I
11
50
35
11
50
35
B
3CJGA_KIM
(KDR)
TK
GW_2580
I
10
43
49
10
43
49
B
1Y6BA_AAX
(KDR)
TK
AAX
I
1
13
1
1
13
1
B
1Y6AA_AAZ
(KDR)
TK
AAZ
I
1
26
1
1
26
1
E
15
3C7QA_XIN
(KDR)
TK
BIBF1120
I
25
56
50
E
3C7QA_XIN
(KDR)
TK
BIBF1120
I
25
56
50
25
56
50
E
3BE2A_RAJ
(KDR)
TK
RAJ
II
19
249
47
19
249
47
E
3EWHA_K11
(KDR)
TK
k11
II
17
27
46
17
27
46
E
1YWNA_LIF
(KDR)
TK
AC1NS1DP
II
17
49
42
17
49
42
E
3EFLA_706
(KDR)
TK
Motesanib
II
15
69
43
15
69
43
E
2P2IA_608
(KDR)
TK
nicotinamide...
II
15
58
45
15
58
45
E
3CPBA_C92
(KDR)
TK
3cpb
II
12
86
32
12
86
32
E
2OH4A_GIG
(KDR)
TK
2oh4
II
9
89
35
9
89
35
E
3DTWA_A96
(KDR)
TK
DB07326
II
8
35
25
8
35
25
E
3CP9A_C19
(KDR)
TK
3cp9
II
6
15
26
6
15
26
E
3B8QA_900
(KDR)
TK
3b8q
II
6
79
20
6
79
20
E
2QU6A_857
(KDR)
TK
2-aminobenzo...
II
5
26
25
5
26
25
E
3CPCA_C52
(KDR)
TK
3cpc
II
5
10
16
5
10
16
E
2QU5A_276
(KDR)
TK
2qu5
II
5
33
25
5
33
25
E
2XIRA_00J
(KDR)
TK
3b8r
I
5
16
24
5
16
24
F
1
2RL5A_2RL
(KDR)
TK
Sorafenib
II
12
94
45
F
2RL5A_2RL
(KDR)
TK
Sorafenib
II
12
94
45
12
94
45