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Diseases
Inhibitor-Anchor Map
Family Anchors
Kinase-Inhibitor Family
Template
Protein
Surface
Ribbon
Inhibitor
ATP Location
Pocket
ATP
NLP
HAP
CLP
SP
1 PRKCE related diseases
hsa04930
Type II diabetes mellitus
Summary of query kinase
Query kinase
PRKCE (
Q02156
)
Kinase group
AGC
Number of conformation types
0
Number of structural templates
39 (
Total 216 inhibitors
)
Number of PRKCE related diseases
1 (
hsa04930
)
Select
Template
Comformation
Type
No. of
Templates
Representative
Template
Kinase
Group
Representative
Inhibitor
Inhibitor
Type
No. of
Kinases
No. of
Inhibitors
No. of
Diseases
A
36
3KRWA_BA1
(ADRBK1)
AGC
balanol
I
17
127
29
A
3KRWA_BA1
(ADRBK1)
AGC
balanol
I
17
127
29
17
127
29
A
1XWSA_BI1
(PIM1)
AGC
bisindolylma...
I
41
132
36
41
132
36
A
2BIKB_BI1
(PIM1)
AGC
bisindolylma...
I
41
132
36
41
132
36
A
2BILB_BI1
(PIM1)
AGC
bisindolylma...
I
41
132
36
41
132
36
A
2I0EA_PDS
(PRKCB)
AGC
bisindolylma...
I
41
141
45
41
141
45
A
3IW4A_LW4
(PRKCA)
AGC
Sotrastaurin
I
52
119
49
52
119
49
A
2OW3A_BIM
(GSK3B)
AGC
LY_333531
I
62
139
51
62
139
51
A
2J2IB_LY4
(PIM1)
AGC
Ruboxistaurin
I
35
89
36
35
89
36
A
1AQ1A_STU
(CDK2)
AGC
staurosporine
I
195
76
118
195
76
118
A
1YHSA_STU
(PIM1)
AGC
staurosporine
I
78
64
50
78
64
50
A
1BYGA_STU
(CSK)
AGC
staurosporine
I
85
72
123
85
72
123
A
2DQ7X_STU
(FYN)
AGC
staurosporine
I
91
74
124
91
74
124
A
1NVQA_UCN
(CHEK1)
AGC
UCN 02
I
179
65
79
179
65
79
A
2HZ4A_4ST
(ABL1)
AGC
staurosporine
I
159
103
156
159
103
156
A
1NVRA_STU
(CHEK1)
AGC
staurosporine
I
179
71
79
179
71
79
A
3A4OX_STU
(LYN)
AGC
staurosporine
I
73
70
88
73
70
88
A
1NXKA_STU
(MAPKAPK2)
AGC
staurosporine
I
110
67
51
110
67
51
A
3CKXA_STU
(STK24)
AGC
staurosporine
I
176
104
141
176
104
141
A
1PKDA_UCN
(CDK2)
AGC
UCN 02
I
195
67
118
195
67
118
A
1Q3DA_STU
(GSK3B)
AGC
staurosporine
I
115
71
61
115
71
61
A
1XJDA_STU
(PRKCQ)
AGC
staurosporine
I
121
101
106
121
101
106
A
3NLBA_5BE
(CHEK1)
AGC
38P
I
45
115
49
45
115
49
A
3EQFA_KSA
(MAP2K1)
AGC
k-252a
I
42
51
57
42
51
57
A
2IW6A_QQ2
(CDK2)
AGC
2iw6
I
112
209
86
112
209
86
A
3BHHA_5CP
(CAMK2B)
AGC
DCL001071
I
17
45
22
17
45
22
A
2CKEA_IQU
(DAPK2)
AGC
AEIQS
I
10
17
22
10
17
22
A
3LM0A_EBD
(STK17B)
AGC
DCL001071
I
20
106
24
20
106
24
A
2JDRA_L20
(AKT2)
AGC
A-443654
I
44
255
61
44
255
61
A
3A2CA_PDY
(MAPKAPK2)
AGC
6-(4-methoxy...
I
32
39
21
32
39
21
A
1NVSA_UCM
(CHEK1)
AGC
SB218078
I
97
6
53
97
6
53
A
2JEDA_LG8
(PRKCQ)
AGC
5-Arylidene-...
I
67
19
87
67
19
87
A
2J51A_DKI
(SLK)
AGC
5-AMINO-3-{[...
I
90
11
103
90
11
103
A
2HY0A_306
(CHEK1)
AGC
AMG_706
I
23
80
49
23
80
49
A
2JFLA_DKI
(SLK)
AGC
5-AMINO-3-{[...
I
90
11
103
90
11
103
A
3D0EA_G93
(AKT2)
AGC
9-N-ethyl-8-...
I
30
15
45
30
15
45
A
2UV2A_GVD
(SLK)
AGC
pyrido[4,3-d...
I
21
80
62
21
80
62
B
3
3D7TA_STU
(CSK)
AGC
staurosporine
I
70
68
99
B
3D7TA_STU
(CSK)
AGC
staurosporine
I
70
68
99
70
68
99
B
1H07A_MFP
(CDK2)
AGC
AC1NAKJQ
I
90
241
80
90
241
80
B
1OIRA_HDY
(CDK2)
AGC
AC1O6YZF
I
51
203
64
51
203
64