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Diseases
Inhibitor-Anchor Map
Family Anchors
Kinase-Inhibitor Family
Template
Protein
Surface
Ribbon
Inhibitor
ATP Location
Pocket
ATP
NLP
HAP
CLP
SP
1 PDPK1 related diseases
hsa05215
Prostate cancer
Summary of query kinase
Query kinase
PDPK1 (
O15530
)
Kinase group
AGC
Number of conformation types
2
Number of structural templates
37 (
Total 229 inhibitors
)
Number of PDPK1 related diseases
1 (
hsa05215
)
Select
Template
Comformation
Type
No. of
Templates
Representative
Template
Kinase
Group
Representative
Inhibitor
Inhibitor
Type
No. of
Kinases
No. of
Inhibitors
No. of
Diseases
A
2
3QC4A_MP7
(PDPK1)
AGC
pyrimidone, 39
II
1
1
1
A
3QC4A_MP7
(PDPK1)
AGC
pyrimidone, 39
II
1
1
1
1
1
1
A
3NAXA_MP7
(PDPK1)
AGC
pyrimidone, 39
II
1
1
1
1
1
1
B
35
1OKYA_STU
(PDPK1)
AGC
staurosporine
I
179
67
109
B
1OKYA_STU
(PDPK1)
AGC
staurosporine
I
179
67
109
179
67
109
B
1OKZA_UCN
(PDPK1)
AGC
UCN 02
I
179
60
109
179
60
109
B
2PE2A_464
(PDPK1)
AGC
Indolinone b...
I
134
156
104
134
156
104
B
1UU8A_BI1
(PDPK1)
AGC
bisindolylma...
I
83
189
65
83
189
65
B
1UU9A_BI3
(PDPK1)
AGC
3-[1-(3-AMIN...
I
83
180
69
83
180
69
B
3OTUA_BI4
(PDPK1)
AGC
bisindolylma...
I
82
178
65
82
178
65
B
1UVRA_BI8
(PDPK1)
AGC
Ro 31-7549
I
82
181
65
82
181
65
B
1UU7A_BI2
(PDPK1)
AGC
bisindolylma...
I
82
178
65
82
178
65
B
3ORZA_BI4
(PDPK1)
AGC
bisindolylma...
I
82
178
65
82
178
65
B
1UU3A_LY4
(PDPK1)
AGC
Ruboxistaurin
I
71
117
57
71
117
57
B
2XCKA_MH4
(PDPK1)
AGC
MH4
I
46
431
75
46
431
75
B
3H9OA_9BD
(PDPK1)
AGC
Benzo[c][2,7...
I
45
68
71
45
68
71
B
3HRFA_ATP
(PDPK1)
AGC
Adenosine-5'...
I
30
9
67
30
9
67
B
3HRCA_ATP
(PDPK1)
AGC
Adenosine-5'...
I
30
9
67
30
9
67
B
1H1WA_ATP
(PDPK1)
AGC
Adenosine-5'...
I
30
9
67
30
9
67
B
2BIYA_ATP
(PDPK1)
AGC
Adenosine-5'...
I
30
9
67
30
9
67
B
3QD0A_3Q4
(PDPK1)
AGC
(3s,6r)-1-[2...
I
28
114
63
28
114
63
B
3QCQA_3Q0
(PDPK1)
AGC
Kinome_1060
I
20
63
45
20
63
45
B
2PE0A_39Z
(PDPK1)
AGC
2pe0
I
20
2
27
20
2
27
B
3NAYA_MP6
(PDPK1)
AGC
ZINC13474643
I
20
81
37
20
81
37
B
2XCHA_CKG
(PDPK1)
AGC
LY_333531
I
19
83
41
19
83
41
B
3IONA_8H1
(PDPK1)
AGC
8H1
I
16
93
51
16
93
51
B
3IOPA_8I1
(PDPK1)
AGC
8H1
I
16
93
51
16
93
51
B
1Z5MA_LI8
(PDPK1)
AGC
BX-320
I
11
35
28
11
35
28
B
3QCSA_3Q1
(PDPK1)
AGC
HMS3303J20
I
7
11
31
7
11
31
B
2R7BA_253
(PDPK1)
AGC
Kinome_3774
I
7
51
23
7
51
23
B
3QCXA_3Q2
(PDPK1)
AGC
HMS3303J20
I
7
11
31
7
11
31
B
3QD4A_3Q6
(PDPK1)
AGC
3Q6
I
5
10
27
5
10
27
B
3QD3A_3Q5
(PDPK1)
AGC
3Q6
I
5
10
27
5
10
27
B
3QCYA_3Q3
(PDPK1)
AGC
(3s,6r)-1-[2...
I
5
13
16
5
13
16
B
3HRFA_P47
(PDPK1)
AGC
(Z)-5-(4-Chl...
I
2
4
14
2
4
14
B
3ORXA_1F8
(PDPK1)
AGC
DNC004786
I
1
1
1
1
1
1
B
2PE1A_517
(PDPK1)
AGC
BX-517
I
1
1
1
1
1
1
B
3PWYA_SYP
(PDPK1)
AGC
CP_690550
I
1
1
1
1
1
1
B
3RCJA_3RC
(PDPK1)
AGC
ZINC00532702
I
1
1
1
1
1
1