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Diseases
Inhibitor-Anchor Map
Family Anchors
Kinase-Inhibitor Family
Template
Protein
Surface
Ribbon
Inhibitor
ATP Location
Pocket
ATP
NLP
HAP
CLP
SP
12 AKT3 related diseases
hsa05142
Chagas disease (American trypanosomiasis)
hsa05145
Toxoplasmosis
hsa05152
Tuberculosis
hsa05160
Hepatitis C
hsa05162
Measles
hsa05164
Influenza A
hsa05169
Epstein-Barr virus infection
hsa05215
Prostate cancer
hsa05218
Melanoma
hsa05220
Chronic myeloid leukemia
hsa05221
Acute myeloid leukemia
hsa05222
Small cell lung cancer
Summary of query kinase
Query kinase
AKT3 (
Q9Y243
)
Kinase group
AGC
Number of conformation types
0
Number of structural templates
52 (
Total 140 inhibitors
)
Number of AKT3 related diseases
12 (
hsa05142
hsa05145
hsa05152
hsa05160
hsa05162
hsa05164
hsa05169
hsa05215
...
)
Select
Template
Comformation
Type
No. of
Templates
Representative
Template
Kinase
Group
Representative
Inhibitor
Inhibitor
Type
No. of
Kinases
No. of
Inhibitors
No. of
Diseases
A
30
2JDRA_L20
(AKT2)
AGC
A-443654
I
44
255
61
A
2JDRA_L20
(AKT2)
AGC
A-443654
I
44
255
61
44
255
61
A
3E87A_G95
(AKT2)
AGC
AG_013736
I
9
42
28
9
42
28
A
2GHGA_A53
(CHEK1)
AGC
oxindole pyr...
I
10
102
25
10
102
25
A
2X39A_X39
(AKT2)
AGC
4-Amino-N-(4...
I
6
93
25
6
93
25
A
1XJDA_STU
(PRKCQ)
AGC
staurosporine
I
121
101
106
121
101
106
A
1BYGA_STU
(CSK)
AGC
staurosporine
I
85
72
123
85
72
123
A
1YHSA_STU
(PIM1)
AGC
staurosporine
I
78
64
50
78
64
50
A
1NVQA_UCN
(CHEK1)
AGC
UCN 02
I
179
65
79
179
65
79
A
1YVJA_4ST
(JAK3)
AGC
staurosporine
I
96
90
126
96
90
126
A
1NVRA_STU
(CHEK1)
AGC
staurosporine
I
179
71
79
179
71
79
A
1PKDA_UCN
(CDK2)
AGC
UCN 02
I
195
67
118
195
67
118
A
1SM2A_STU
(ITK)
AGC
staurosporine
I
99
104
128
99
104
128
A
1SNUA_STU
(ITK)
AGC
staurosporine
I
99
104
128
99
104
128
A
1AQ1A_STU
(CDK2)
AGC
staurosporine
I
195
76
118
195
76
118
A
3IW4A_LW4
(PRKCA)
AGC
Sotrastaurin
I
52
119
49
52
119
49
A
1XWSA_BI1
(PIM1)
AGC
bisindolylma...
I
41
132
36
41
132
36
A
3E88A_G96
(AKT2)
AGC
ZSGNCHLJBWLF...
I
3
16
20
3
16
20
A
3E8DA_G98
(AKT2)
AGC
Roscovitine
I
5
19
21
5
19
21
A
2BIKB_BI1
(PIM1)
AGC
bisindolylma...
I
41
132
36
41
132
36
A
2BILB_BI1
(PIM1)
AGC
bisindolylma...
I
41
132
36
41
132
36
A
2I0EA_PDS
(PRKCB)
AGC
bisindolylma...
I
41
141
45
41
141
45
A
2J2IB_LY4
(PIM1)
AGC
Ruboxistaurin
I
35
89
36
35
89
36
A
3NLBA_5BE
(CHEK1)
AGC
38P
I
45
115
49
45
115
49
A
2B55A_D31
(CDK2)
AGC
D31
I
27
87
53
27
87
53
A
3D0EA_G93
(AKT2)
AGC
9-N-ethyl-8-...
I
30
15
45
30
15
45
A
2E9VA_85A
(CHEK1)
AGC
macrocyclic ...
I
14
121
27
14
121
27
A
2HXQA_373
(CHEK1)
AGC
DB07025
I
7
36
26
7
36
26
A
2HY0A_306
(CHEK1)
AGC
AMG_706
I
23
80
49
23
80
49
A
1NVSA_UCM
(CHEK1)
AGC
SB218078
I
97
6
53
97
6
53
A
2JDOA_I5S
(AKT2)
AGC
I5S
I
10
22
29
10
22
29
B
22
2GU8A_796
(PRKACA)
AGC
DB07235
I
7
38
29
B
2GU8A_796
(PRKACA)
AGC
DB07235
I
7
38
29
7
38
29
B
3OCBA_XM1
(AKT1)
AGC
XM1
I
10
99
23
10
99
23
B
3BKBA_STU
(FES)
AGC
staurosporine
I
131
107
138
131
107
138
B
1OKYA_STU
(PDPK1)
AGC
staurosporine
I
179
67
109
179
67
109
B
3CBLA_STU
(FES)
AGC
staurosporine
I
131
107
138
131
107
138
B
1OKZA_UCN
(PDPK1)
AGC
UCN 02
I
179
60
109
179
60
109
B
3CD3A_STU
(FES)
AGC
staurosporine
I
131
107
138
131
107
138
B
3MVHA_WFE
(AKT1)
AGC
N-{[(3s)-3-A...
I
5
44
23
5
44
23
B
3OW4A_SMY
(AKT1)
AGC
LY_317615
I
3
37
20
3
37
20
B
1UU9A_BI3
(PDPK1)
AGC
3-[1-(3-AMIN...
I
83
180
69
83
180
69
B
1UVRA_BI8
(PDPK1)
AGC
Ro 31-7549
I
82
181
65
82
181
65
B
3ORZA_BI4
(PDPK1)
AGC
bisindolylma...
I
82
178
65
82
178
65
B
3OTUA_BI4
(PDPK1)
AGC
bisindolylma...
I
82
178
65
82
178
65
B
1ZRZA_BI1
(PRKCI)
AGC
bisindolylma...
I
52
150
47
52
150
47
B
1UU7A_BI2
(PDPK1)
AGC
bisindolylma...
I
82
178
65
82
178
65
B
1UU8A_BI1
(PDPK1)
AGC
bisindolylma...
I
83
189
65
83
189
65
B
2XCHA_CKG
(PDPK1)
AGC
LY_333531
I
19
83
41
19
83
41
B
1UU3A_LY4
(PDPK1)
AGC
Ruboxistaurin
I
71
117
57
71
117
57
B
3IONA_8H1
(PDPK1)
AGC
8H1
I
16
93
51
16
93
51
B
3IOPA_8I1
(PDPK1)
AGC
8H1
I
16
93
51
16
93
51
B
3QD0A_3Q4
(PDPK1)
AGC
(3s,6r)-1-[2...
I
28
114
63
28
114
63
B
3L9MA_L9M
(PRKACA)
AGC
VX_680
I
37
65
42
37
65
42