|
Query kinase |
AURKB (Q96GD4)
|
Kinase group |
Other |
Number of conformation types |
0 |
Number of structural templates |
197 (Total 596 inhibitors) |
Select Template |
Comformation Type |
No. of Templates |
Representative Template |
Kinase Group |
Representative Inhibitor |
Inhibitor Type |
No. of Kinases |
No. of Inhibitors |
No. of Diseases |
|
A |
105
|
2F4JA_VX6 (ABL1) |
Other |
VX-680 |
I |
110 |
109
| 134 |
|
|
B |
92
|
2C6EA_HPM (AURKA) |
Other |
HPM |
I |
44 |
237
| 90 |
|
B |
2C6EA_HPM (AURKA) |
Other |
HPM |
I |
44 |
237 |
90 |
44 |
237 |
90 |
|
B |
2PE2A_464 (PDPK1) |
Other |
Indolinone b... |
I |
134 |
156 |
104 |
134 |
156 |
104 |
|
B |
3H10A_97B (AURKA) |
Other |
MLN8054 |
I |
39 |
88 |
82 |
39 |
88 |
82 |
|
B |
3DA6A_BZ9 (MAPK10) |
Other |
BZ9 |
I |
5 |
26 |
17 |
5 |
26 |
17 |
|
B |
2XCKA_MH4 (PDPK1) |
Other |
MH4 |
I |
46 |
431 |
75 |
46 |
431 |
75 |
|
B |
3EFWA_AK8 (AURKA) |
Other |
3efw |
I |
100 |
59 |
105 |
100 |
59 |
105 |
|
B |
3MYGA_EML (AURKA) |
Other |
Roscovitine |
I |
6 |
23 |
12 |
6 |
23 |
12 |
|
B |
2XRUA_400 (AURKA) |
Other |
VX_680 |
I |
33 |
152 |
63 |
33 |
152 |
63 |
|
B |
3NRMA_NRM (AURKA) |
Other |
CAS404828_08_6 |
I |
32 |
33 |
60 |
32 |
33 |
60 |
|
B |
2W1EA_L0E (AURKA) |
Other |
pyrazole-ben... |
I |
15 |
32 |
45 |
15 |
32 |
45 |
|
B |
3CBLA_STU (FES) |
Other |
staurosporine |
I |
131 |
107 |
138 |
131 |
107 |
138 |
|
B |
2J4ZA_626 (AURKA) |
Other |
2j4z |
I |
13 |
51 |
25 |
13 |
51 |
25 |
|
B |
2BMCA_MPY (AURKA) |
Other |
PHA-680632 |
I |
107 |
108 |
107 |
107 |
108 |
107 |
|
B |
3CD3A_STU (FES) |
Other |
staurosporine |
I |
131 |
107 |
138 |
131 |
107 |
138 |
|
B |
1WVYA_STU (DAPK1) |
Other |
staurosporine |
I |
83 |
23 |
55 |
83 |
23 |
55 |
|
B |
3LCSA_STU (ALK) |
Other |
staurosporine |
I |
73 |
100 |
109 |
73 |
100 |
109 |
|
B |
1OKYA_STU (PDPK1) |
Other |
staurosporine |
I |
179 |
67 |
109 |
179 |
67 |
109 |
|
B |
3MIYA_B49 (ITK) |
Other |
Sunitinib |
I |
70 |
74 |
110 |
70 |
74 |
110 |
|
B |
3BKBA_STU (FES) |
Other |
staurosporine |
I |
131 |
107 |
138 |
131 |
107 |
138 |
|
B |
1OKZA_UCN (PDPK1) |
Other |
UCN 02 |
I |
179 |
60 |
109 |
179 |
60 |
109 |
|
B |
2W1GA_L0G (AURKA) |
Other |
AT9283 |
I |
8 |
18 |
21 |
8 |
18 |
21 |
|
B |
2W1IA_L0I (JAK2) |
Other |
AT9283 |
I |
7 |
13 |
21 |
7 |
13 |
21 |
|
B |
1PXPA_CK8 (CDK2) |
Other |
CK8 |
I |
14 |
49 |
26 |
14 |
49 |
26 |
|
B |
1PXNA_CK6 (CDK2) |
Other |
CK6 |
I |
9 |
22 |
14 |
9 |
22 |
14 |
|
B |
1UNHA_IXM (CDK5) |
Other |
INDIRUBIN-3'... |
I |
8 |
25 |
10 |
8 |
25 |
10 |
|
B |
3COHA_83H (AURKA) |
Other |
AKI-001 |
I |
79 |
88 |
65 |
79 |
88 |
65 |
|
B |
3QD0A_3Q4 (PDPK1) |
Other |
(3s,6r)-1-[2... |
I |
28 |
114 |
63 |
28 |
114 |
63 |
|
B |
2WTWA_ZZL (AURKA) |
Other |
MLN8054 |
I |
35 |
24 |
70 |
35 |
24 |
70 |
|
B |
1OIQA_HDU (CDK2) |
Other |
AC1L9L2U |
I |
14 |
56 |
31 |
14 |
56 |
31 |
|
B |
2XA4A_AZ5 (JAK2) |
Other |
AZD1480, AZ... |
I |
15 |
85 |
58 |
15 |
85 |
58 |
|
B |
2J50A_627 (AURKA) |
Other |
5-Amido-pyrr... |
I |
11 |
19 |
34 |
11 |
19 |
34 |
|
B |
3IOKA_1P6 (JAK2) |
Other |
PTK_787 |
I |
16 |
98 |
47 |
16 |
98 |
47 |
|
B |
3AMAA_SKE (PRKACA) |
Other |
JNJ-7706621 |
I |
46 |
26 |
35 |
46 |
26 |
35 |
|
B |
3O2MA_46A (MAPK8) |
Other |
tetrazolylyp... |
I |
11 |
21 |
27 |
11 |
21 |
27 |
|
B |
1PXMA_CK5 (CDK2) |
Other |
CK5 |
I |
12 |
36 |
19 |
12 |
36 |
19 |
|
B |
2R3HA_SCE (CDK2) |
Other |
benzimidazoq... |
I |
15 |
40 |
39 |
15 |
40 |
39 |
|
B |
2W1CA_L0C (AURKA) |
Other |
pyrazole-ben... |
I |
7 |
10 |
28 |
7 |
10 |
28 |
|
B |
3QCQA_3Q0 (PDPK1) |
Other |
Kinome_1060 |
I |
20 |
63 |
45 |
20 |
63 |
45 |
|
B |
1JVPP_LIG (CDK2) |
Other |
ellipticine |
I |
17 |
30 |
45 |
17 |
30 |
45 |
|
B |
3H9OA_9BD (PDPK1) |
Other |
Benzo[c][2,7... |
I |
45 |
68 |
71 |
45 |
68 |
71 |
|
B |
2R3GA_SC9 (CDK2) |
Other |
2r3j |
I |
30 |
137 |
50 |
30 |
137 |
50 |
|
B |
3H0ZA_45B (AURKA) |
Other |
2,4-Bisanili... |
I |
12 |
60 |
44 |
12 |
60 |
44 |
|
B |
2X4FA_16X (MYLK4) |
Other |
AC1O6ZEW |
I |
3 |
5 |
1 |
3 |
5 |
1 |
|
B |
2EXMA_ZIP (CDK2) |
Other |
MLS000079197 |
I |
12 |
22 |
32 |
12 |
22 |
32 |
|
B |
3H0YA_48B (AURKA) |
Other |
2,4-Bisanili... |
I |
7 |
24 |
26 |
7 |
24 |
26 |
|
B |
1PXLA_CK4 (CDK2) |
Other |
4-(2,4-DIMET... |
I |
11 |
22 |
18 |
11 |
22 |
18 |
|
B |
1PF8A_SU9 (CDK2) |
Other |
SU 9516 |
I |
25 |
19 |
33 |
25 |
19 |
33 |
|
B |
2W1DA_L0D (AURKA) |
Other |
AC1NTGE7 |
I |
21 |
31 |
54 |
21 |
31 |
54 |
|
B |
2X6EA_YM4 (AURKA) |
Other |
6-Bromo-7-{4... |
I |
4 |
36 |
3 |
4 |
36 |
3 |
|
B |
3PY0A_SU9 (CDK2) |
Other |
SU 9516 |
I |
25 |
19 |
33 |
25 |
19 |
33 |
|
B |
3PY1A_SU9 (CDK2) |
Other |
SU 9516 |
I |
25 |
19 |
33 |
25 |
19 |
33 |
|
B |
1Z5MA_LI8 (PDPK1) |
Other |
BX-320 |
I |
11 |
35 |
28 |
11 |
35 |
28 |
|
B |
2W1FA_L0F (AURKA) |
Other |
DB08066 |
I |
17 |
40 |
35 |
17 |
40 |
35 |
|
B |
2B1PA_AIZ (MAPK10) |
Other |
AIZ |
I |
7 |
43 |
17 |
7 |
43 |
17 |
|
B |
2W1HA_L0H (CDK2) |
Other |
DB08066 |
I |
20 |
43 |
42 |
20 |
43 |
42 |
|
B |
3NYNA_SGV (GRK6) |
Other |
SMR000127424 |
I |
54 |
7 |
47 |
54 |
7 |
47 |
|
B |
3L9NA_L9N (PRKACA) |
Other |
A_674563 |
I |
10 |
63 |
36 |
10 |
63 |
36 |
|
B |
2C68A_CT6 (CDK2) |
Other |
2c68 |
I |
23 |
73 |
43 |
23 |
73 |
43 |
|
B |
3QD3A_3Q5 (PDPK1) |
Other |
3Q6 |
I |
5 |
10 |
27 |
5 |
10 |
27 |
|
B |
1URWA_I1P (CDK2) |
Other |
Imidazo[1,2-... |
I |
12 |
73 |
29 |
12 |
73 |
29 |
|
B |
2PE0A_39Z (PDPK1) |
Other |
2pe0 |
I |
20 |
2 |
27 |
20 |
2 |
27 |
|
B |
2C6OA_4SP (CDK2) |
Other |
nu6102 |
I |
23 |
33 |
27 |
23 |
33 |
27 |
|
B |
2VZ6A_FEF (CAMK2A) |
Other |
indirubin de... |
I |
15 |
3 |
14 |
15 |
3 |
14 |
|
B |
2C69A_CT8 (CDK2) |
Other |
CT8 |
I |
22 |
62 |
38 |
22 |
62 |
38 |
|
B |
3QD4A_3Q6 (PDPK1) |
Other |
3Q6 |
I |
5 |
10 |
27 |
5 |
10 |
27 |
|
B |
2R64A_740 (CDK2) |
Other |
2r64 |
I |
5 |
27 |
11 |
5 |
27 |
11 |
|
B |
2R3IA_SCF (CDK2) |
Other |
2c68 |
I |
23 |
89 |
43 |
23 |
89 |
43 |
|
B |
2R3JA_SCJ (CDK2) |
Other |
2r3j |
I |
27 |
99 |
49 |
27 |
99 |
49 |
|
B |
1UNLA_RRC (CDK5) |
Other |
roscovitine |
I |
45 |
237 |
47 |
45 |
237 |
47 |
|
B |
3PTGA_932 (MAPK10) |
Other |
N-[4-Methyl-... |
I |
5 |
19 |
15 |
5 |
19 |
15 |
|
B |
1PXOA_CK7 (CDK2) |
Other |
CK7 |
I |
9 |
23 |
17 |
9 |
23 |
17 |
|
B |
1KE5A_LS1 (CDK2) |
Other |
LS1 |
I |
5 |
31 |
6 |
5 |
31 |
6 |
|
B |
2R3FA_SC8 (CDK2) |
Other |
2c68 |
I |
22 |
62 |
43 |
22 |
62 |
43 |
|
B |
2R3KA_SCQ (CDK2) |
Other |
2r3j |
I |
28 |
95 |
49 |
28 |
95 |
49 |
|
B |
2A4LA_RRC (CDK2) |
Other |
roscovitine |
I |
50 |
240 |
50 |
50 |
240 |
50 |
|
B |
2B7AA_IZA (JAK2) |
Other |
Pyridone 6 |
I |
34 |
12 |
65 |
34 |
12 |
65 |
|
B |
3Q32A_J2I (JAK2) |
Other |
2-(2,6-Diflu... |
I |
4 |
29 |
18 |
4 |
29 |
18 |
|
B |
1KE9A_LS5 (CDK2) |
Other |
LS5 |
I |
5 |
27 |
6 |
5 |
27 |
6 |
|
B |
3E63A_5B2 (JAK2) |
Other |
5-phenyl-1H-... |
I |
15 |
29 |
39 |
15 |
29 |
39 |
|
B |
3DDQA_RRC (CDK2) |
Other |
roscovitine |
I |
50 |
240 |
50 |
50 |
240 |
50 |
|
B |
2XB7A_GUI (ALK) |
Other |
NVP-TAE684 |
I |
71 |
66 |
107 |
71 |
66 |
107 |
|
B |
3L9MA_L9M (PRKACA) |
Other |
VX_680 |
I |
37 |
65 |
42 |
37 |
65 |
42 |
|
B |
3CGOA_JNO (MAPK10) |
Other |
DB08026 |
I |
13 |
32 |
21 |
13 |
32 |
21 |
|
B |
1DI8A_DTQ (CDK2) |
Other |
whi-p180 |
I |
26 |
68 |
46 |
26 |
68 |
46 |
|
B |
3P9JA_P9J (AURKA) |
Other |
4-[(5-Methyl... |
I |
32 |
50 |
54 |
32 |
50 |
54 |
|
B |
3IO7A_1P5 (JAK2) |
Other |
CP_690550 |
I |
24 |
65 |
60 |
24 |
65 |
60 |
|
B |
3PJ8A_404 (CDK2) |
Other |
imidazo[2,1-... |
I |
47 |
223 |
49 |
47 |
223 |
49 |
|
B |
2O2UA_738 (MAPK10) |
Other |
2-[(2-chloro... |
I |
9 |
19 |
21 |
9 |
19 |
21 |
|
B |
3M11A_AKI (AURKA) |
Other |
1-(4-{2-[(5,... |
I |
8 |
29 |
27 |
8 |
29 |
27 |
|
B |
3QCYA_3Q3 (PDPK1) |
Other |
(3s,6r)-1-[2... |
I |
5 |
13 |
16 |
5 |
13 |
16 |
|
B |
2C6IA_DT1 (CDK2) |
Other |
2c6i |
I |
27 |
41 |
48 |
27 |
41 |
48 |
|
B |
2VTAA_LZ1 (CDK2) |
Other |
1H-Indazole |
I |
7 |
3 |
26 |
7 |
3 |
26 |
|
|