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Diseases
Inhibitor-Anchor Map
Family Anchors
Kinase-Inhibitor Family
Template
Protein
Surface
Ribbon
Inhibitor
ATP Location
Pocket
ATP
NLP
HAP
CLP
SP
1 PKN1 related diseases
hsa05132
Salmonella infection
Summary of query kinase
Query kinase
PKN1 (
Q16512
)
Kinase group
AGC
Number of conformation types
0
Number of structural templates
49 (
Total 65 inhibitors
)
Number of PKN1 related diseases
1 (
hsa05132
)
Select
Template
Comformation
Type
No. of
Templates
Representative
Template
Kinase
Group
Representative
Inhibitor
Inhibitor
Type
No. of
Kinases
No. of
Inhibitors
No. of
Diseases
A
43
1BYGA_STU
(CSK)
AGC
staurosporine
I
85
72
123
A
1BYGA_STU
(CSK)
AGC
staurosporine
I
85
72
123
85
72
123
A
1XJDA_STU
(PRKCQ)
AGC
staurosporine
I
121
101
106
121
101
106
A
1YVJA_4ST
(JAK3)
AGC
staurosporine
I
96
90
126
96
90
126
A
1NVRA_STU
(CHEK1)
AGC
staurosporine
I
179
71
79
179
71
79
A
2DQ7X_STU
(FYN)
AGC
staurosporine
I
91
74
124
91
74
124
A
1NXKA_STU
(MAPKAPK2)
AGC
staurosporine
I
110
67
51
110
67
51
A
2HZ4A_4ST
(ABL1)
AGC
staurosporine
I
159
103
156
159
103
156
A
3A4OX_STU
(LYN)
AGC
staurosporine
I
73
70
88
73
70
88
A
1QPDA_STU
(LCK)
AGC
staurosporine
I
115
76
126
115
76
126
A
3CKXA_STU
(STK24)
AGC
staurosporine
I
176
104
141
176
104
141
A
1QPJA_STU
(LCK)
AGC
staurosporine
I
115
76
126
115
76
126
A
1AQ1A_STU
(CDK2)
AGC
staurosporine
I
195
76
118
195
76
118
A
1U59A_STU
(ZAP70)
AGC
staurosporine
I
96
80
114
96
80
114
A
1NVQA_UCN
(CHEK1)
AGC
UCN 02
I
179
65
79
179
65
79
A
1PKDA_UCN
(CDK2)
AGC
UCN 02
I
195
67
118
195
67
118
A
2I0EA_PDS
(PRKCB)
AGC
bisindolylma...
I
41
141
45
41
141
45
A
3IW4A_LW4
(PRKCA)
AGC
Sotrastaurin
I
52
119
49
52
119
49
A
2VTTA_LZD
(CDK2)
AGC
pyrazole dia...
I
158
42
111
158
42
111
A
3M2WA_L8I
(MAPKAPK2)
AGC
Sunitinib
I
84
90
47
84
90
47
A
2F4JA_VX6
(ABL1)
AGC
VX-680
I
110
109
134
110
109
134
A
2WIHA_P48
(CDK2)
AGC
VX_680
I
111
425
105
111
425
105
A
2XYNA_VX6
(ABL2)
AGC
VX-680
I
79
101
105
79
101
105
A
3E5AA_VX6
(AURKA)
AGC
VX-680
I
57
107
93
57
107
93
A
3EQFA_KSA
(MAP2K1)
AGC
k-252a
I
42
51
57
42
51
57
A
1R78A_FMD
(CDK2)
AGC
4-alkynyl ox...
I
127
24
97
127
24
97
A
2CKEA_IQU
(DAPK2)
AGC
AEIQS
I
10
17
22
10
17
22
A
1NVSA_UCM
(CHEK1)
AGC
SB218078
I
97
6
53
97
6
53
A
2IW6A_QQ2
(CDK2)
AGC
2iw6
I
112
209
86
112
209
86
A
3NLBA_5BE
(CHEK1)
AGC
38P
I
45
115
49
45
115
49
A
2HOGA_710
(CHEK1)
AGC
3-(Indol-2-y...
I
33
66
51
33
66
51
A
2J51A_DKI
(SLK)
AGC
5-AMINO-3-{[...
I
90
11
103
90
11
103
A
3EIDA_PO5
(CDK2)
AGC
AC1O6YZF
I
63
211
77
63
211
77
A
2JFLA_DKI
(SLK)
AGC
5-AMINO-3-{[...
I
90
11
103
90
11
103
A
3D0EA_G93
(AKT2)
AGC
9-N-ethyl-8-...
I
30
15
45
30
15
45
A
3PJ3A_04L
(BTK)
AGC
Imatinib
II
99
113
134
99
113
134
A
2JDRA_L20
(AKT2)
AGC
A-443654
I
44
255
61
44
255
61
A
1AGWA_SU2
(FGFR1)
AGC
SU 4984
I
77
81
111
77
81
111
A
2J90A_IZA
(DAPK3)
AGC
Pyridone 6
I
40
50
42
40
50
42
A
3PIYA_585
(BTK)
AGC
R-406
I
93
17
123
93
17
123
A
2JEDA_LG8
(PRKCQ)
AGC
5-Arylidene-...
I
67
19
87
67
19
87
A
3LXLA_IZA
(JAK3)
AGC
Pyridone 6
I
30
11
63
30
11
63
A
2JDOA_I5S
(AKT2)
AGC
I5S
I
10
22
29
10
22
29
A
2IVUA_ZD6
(RET)
AGC
Vandetanib
I
83
291
121
83
291
121
B
6
3D7TA_STU
(CSK)
AGC
staurosporine
I
70
68
99
B
3D7TA_STU
(CSK)
AGC
staurosporine
I
70
68
99
70
68
99
B
3FUPA_MI1
(JAK2)
AGC
CP690550
I
16
27
32
16
27
32
B
1OIRA_HDY
(CDK2)
AGC
AC1O6YZF
I
51
203
64
51
203
64
B
2B7AA_IZA
(JAK2)
AGC
Pyridone 6
I
34
12
65
34
12
65
B
1H07A_MFP
(CDK2)
AGC
AC1NAKJQ
I
90
241
80
90
241
80
B
3MTLA_FEF
(PCTK1)
AGC
indirubin de...
I
16
3
23
16
3
23