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Diseases
Inhibitor-Anchor Map
Family Anchors
Kinase-Inhibitor Family
Template
Protein
Surface
Ribbon
Inhibitor
ATP Location
Pocket
ATP
NLP
HAP
CLP
SP
Summary of query kinase
Query kinase
CHEK1 (
O14757
)
Kinase group
CAMK
Number of conformation types
1
Number of structural templates
58 (
Total 1185 inhibitors
)
Select
Template
Comformation
Type
No. of
Templates
Representative
Template
Kinase
Group
Representative
Inhibitor
Inhibitor
Type
No. of
Kinases
No. of
Inhibitors
No. of
Diseases
A
58
1NVQA_UCN
(CHEK1)
CAMK
UCN 02
I
179
65
79
A
1NVQA_UCN
(CHEK1)
CAMK
UCN 02
I
179
65
79
179
65
79
A
1NVRA_STU
(CHEK1)
CAMK
staurosporine
I
179
71
79
179
71
79
A
1NVSA_UCM
(CHEK1)
CAMK
SB218078
I
97
6
53
97
6
53
A
3NLBA_5BE
(CHEK1)
CAMK
38P
I
45
115
49
45
115
49
A
2HOGA_710
(CHEK1)
CAMK
3-(Indol-2-y...
I
33
66
51
33
66
51
A
1ZYSA_199
(CHEK1)
CAMK
2,4-Diamino-...
I
31
92
52
31
92
52
A
2BRNA_DF1
(CHEK1)
CAMK
pyrrolopyrim...
I
30
119
42
30
119
42
A
2BROA_DF2
(CHEK1)
CAMK
pyrrolopyrim...
I
29
109
40
29
109
40
A
2HY0A_306
(CHEK1)
CAMK
AMG_706
I
23
80
49
23
80
49
A
2BRMA_DFZ
(CHEK1)
CAMK
DFZ
I
21
88
36
21
88
36
A
2BRGA_DFY
(CHEK1)
CAMK
DFY
I
18
33
32
18
33
32
A
2E9NA_76A
(CHEK1)
CAMK
2e9n
I
18
39
40
18
39
40
A
2XEZA_XEZ
(CHEK1)
CAMK
CAS396129_53_6
I
16
35
37
16
35
37
A
2C3KA_ABO
(CHEK1)
CAMK
ABO
I
15
47
31
15
47
31
A
1ZLTA_HYM
(CHEK1)
CAMK
10E-Hymenial...
I
15
31
31
15
31
31
A
3PA5A_C73
(CHEK1)
CAMK
2-(Carbamoyl...
I
15
74
20
15
74
20
A
2HXLA_422
(CHEK1)
CAMK
DB07075
I
15
95
36
15
95
36
A
2C3LA_IDZ
(CHEK1)
CAMK
IDZ
I
14
36
26
14
36
26
A
3OT8A_MI5
(CHEK1)
CAMK
VX_680
I
14
63
25
14
63
25
A
2C3JA_DBQ
(CHEK1)
CAMK
Debromohymen...
I
14
33
31
14
33
31
A
2E9VA_85A
(CHEK1)
CAMK
macrocyclic ...
I
14
121
27
14
121
27
A
2XEYA_YVQ
(CHEK1)
CAMK
3-(Indol-2-y...
I
13
35
26
13
35
26
A
3OT3A_22K
(CHEK1)
CAMK
INCB18424
I
13
30
13
13
30
13
A
2XF0A_4UB
(CHEK1)
CAMK
AC1LCX0J
I
12
32
26
12
32
26
A
3PA3A_C70
(CHEK1)
CAMK
2-(4-Chlorop...
I
11
72
16
11
72
16
A
2GHGA_A53
(CHEK1)
CAMK
oxindole pyr...
I
10
102
25
10
102
25
A
3PA4A_C72
(CHEK1)
CAMK
2-(4-Chlorop...
I
10
79
24
10
79
24
A
2BRBA_PFQ
(CHEK1)
CAMK
2-[(5,6-DIPH...
I
8
32
23
8
32
23
A
2HXQA_373
(CHEK1)
CAMK
DB07025
I
7
36
26
7
36
26
A
2WMVA_ZYV
(CHEK1)
CAMK
purine, 10
I
6
18
23
6
18
23
A
2QHNA_582
(CHEK1)
CAMK
AOBLVMINLZGC...
I
6
12
10
6
12
10
A
2BR1A_PFP
(CHEK1)
CAMK
PFP
I
6
11
14
6
11
14
A
2BRHA_DFW
(CHEK1)
CAMK
DFW
I
6
12
19
6
12
19
A
2E9OA_A58
(CHEK1)
CAMK
DB07320
I
6
38
15
6
38
15
A
2WMUA_ZYU
(CHEK1)
CAMK
4-(9h-purin-...
I
6
17
19
6
17
19
A
2WMXA_ZY6
(CHEK1)
CAMK
pyrazolopyri...
I
5
15
22
5
15
22
A
2X8IA_X8I
(CHEK1)
CAMK
PI_103
I
4
19
13
4
19
13
A
2GDOA_12C
(CHEK1)
CAMK
DB06852
I
4
27
17
4
27
17
A
2X8EA_X8E
(CHEK1)
CAMK
CAS318480_82_9
I
4
31
16
4
31
16
A
3JVRA_AGX
(CHEK1)
CAMK
CAS269390_69_4
I
3
5
12
3
5
12
A
2AYPA_43A
(CHEK1)
CAMK
43A
I
3
22
13
3
22
13
A
2WMQA_ZYQ
(CHEK1)
CAMK
AC1LEOLN
I
3
2
6
3
2
6
A
3F9NA_38M
(CHEK1)
CAMK
Sunitinib
I
3
9
16
3
9
16
A
2CGXA_3D3
(CHEK1)
CAMK
2-[(6-amino-...
I
2
2
0
2
2
0
A
2WMSA_ZYS
(CHEK1)
CAMK
ZINC01398629
I
2
2
6
2
2
6
A
2E9UA_A25
(CHEK1)
CAMK
macrocyclic ...
I
2
79
12
2
79
12
A
2WMRA_ZYR
(CHEK1)
CAMK
14346-24-8
I
2
2
3
2
2
3
A
2WMWA_ZYW
(CHEK1)
CAMK
pyrazolopyri...
I
2
8
4
2
8
4
A
2E9PA_77A
(CHEK1)
CAMK
macrocyclic ...
I
1
81
0
1
81
0
A
2CGUA_3A3
(CHEK1)
CAMK
ChemDiv1_019...
I
1
1
0
1
1
0
A
2CGVA_3B3
(CHEK1)
CAMK
3B3
I
1
1
0
1
1
0
A
2CGWA_3C3
(CHEK1)
CAMK
3C3
I
1
1
0
1
1
0
A
2QHMA_7CS
(CHEK1)
CAMK
pyrimidine d...
I
1
1
0
1
1
0
A
3JVSA_AGY
(CHEK1)
CAMK
AC1NWTCI
I
1
1
0
1
1
0
A
2X8DA_X8D
(CHEK1)
CAMK
MLS000085512
I
1
14
0
1
14
0
A
2YWPA_A42
(CHEK1)
CAMK
2ywp
I
1
108
0
1
108
0
A
2R0UA_M54
(CHEK1)
CAMK
M54
I
1
19
0
1
19
0
A
2WMTA_ZYT
(CHEK1)
CAMK
triazole, 4b
I
1
1
0
1
1
0