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Diseases
Inhibitor-Anchor Map
Family Anchors
Kinase-Inhibitor Family
Template
Protein
Surface
Ribbon
Inhibitor
ATP Location
Pocket
ATP
NLP
HAP
CLP
SP
12 MAPK14 related diseases
hsa05014
Amyotrophic lateral sclerosis (ALS)
hsa05120
Epithelial cell signaling in Helicobacter pylori infection
hsa05131
Shigellosis
hsa05132
Salmonella infection
hsa05133
Pertussis
hsa05140
Leishmaniasis
hsa05142
Chagas disease (American trypanosomiasis)
hsa05145
Toxoplasmosis
hsa05152
Tuberculosis
hsa05160
Hepatitis C
hsa05164
Influenza A
hsa05169
Epstein-Barr virus infection
Summary of query kinase
Query kinase
MAPK14 (
Q16539
)
Kinase group
CMGC
Number of conformation types
3
Number of structural templates
119 (
Total 2764 inhibitors
)
Number of MAPK14 related diseases
12 (
hsa05014
hsa05120
hsa05131
hsa05132
hsa05133
hsa05140
hsa05142
hsa05145
...
)
Select
Template
Comformation
Type
No. of
Templates
Representative
Template
Kinase
Group
Representative
Inhibitor
Inhibitor
Type
No. of
Kinases
No. of
Inhibitors
No. of
Diseases
A
75
3L8XA_N4D
(MAPK14)
CMGC
3cg2
I
91
104
65
A
3L8XA_N4D
(MAPK14)
CMGC
3cg2
I
91
104
65
91
104
65
A
3HA8A_5JZ
(MAPK14)
CMGC
DEL-B, 14b
I
59
89
62
59
89
62
A
3IPHA_G11
(MAPK14)
CMGC
HMS3303K05
I
57
108
55
57
108
55
A
3E92A_G6A
(MAPK14)
CMGC
3e92
I
56
59
55
56
59
55
A
2ZB1A_GK4
(MAPK14)
CMGC
biphenyl ami...
II
55
57
54
55
57
54
A
3MVLA_38P
(MAPK14)
CMGC
38P
I
50
308
44
50
308
44
A
1BL6A_SB6
(MAPK14)
CMGC
sb216995
I
46
110
50
46
110
50
A
1ZZLA_TZY
(MAPK14)
CMGC
CP-808844
I
36
84
44
36
84
44
A
1OUKA_084
(MAPK14)
CMGC
1ouk
I
24
139
46
24
139
46
A
3MVMA_39P
(MAPK14)
CMGC
39P
I
24
247
38
24
247
38
A
1BL7A_SB4
(MAPK14)
CMGC
SB220025
I
22
159
29
22
159
29
A
3OBGA_SB2
(MAPK14)
CMGC
SB 203580
I
21
31
28
21
31
28
A
3DS6A_A17
(MAPK14)
CMGC
3ds6
II
21
146
34
21
146
34
A
1A9UA_SB2
(MAPK14)
CMGC
SB 203580
I
21
31
28
21
31
28
A
3BV2A_P38
(MAPK14)
CMGC
MLN_518
II
20
142
37
20
142
37
A
1YQJA_6NP
(MAPK14)
CMGC
AMG_706
I
19
102
43
19
102
43
A
1OZ1A_FPH
(MAPK14)
CMGC
4-Azaindole 6
I
18
27
28
18
27
28
A
3DT1A_P40
(MAPK14)
CMGC
DB08351
II
18
69
32
18
69
32
A
3FKOA_FKO
(MAPK14)
CMGC
L-779450
I
17
7
27
17
7
27
A
3ITZA_P66
(MAPK14)
CMGC
P66
II
15
102
25
15
102
25
A
1BMKA_SB5
(MAPK14)
CMGC
SB-218655
I
14
116
34
14
116
34
A
1DI9A_MSQ
(MAPK14)
CMGC
MSQ
I
14
29
29
14
29
29
A
3FC1X_52P
(MAPK14)
CMGC
VX-745
I
12
6
21
12
6
21
A
3HP5A_52P
(MAPK14)
CMGC
VX-745
I
12
6
21
12
6
21
A
3GFEA_P37
(MAPK14)
CMGC
DB08349
I
11
83
29
11
83
29
A
3FLYA_FLY
(MAPK14)
CMGC
HMS3401N11
I
10
44
29
10
44
29
A
3FLZA_FLZ
(MAPK14)
CMGC
HMS3401P11
I
10
31
23
10
31
23
A
3FMKA_FMK
(MAPK14)
CMGC
FMK
I
10
25
29
10
25
29
A
3FMHA_533
(MAPK14)
CMGC
FMK
I
10
25
29
10
25
29
A
3FKLA_FKL
(MAPK14)
CMGC
38P
I
9
65
23
9
65
23
A
3FSFA_FSS
(MAPK14)
CMGC
AST_487
I
9
52
40
9
52
40
A
3FLNC_3FN
(MAPK14)
CMGC
Kinome_3762
I
9
44
22
9
44
22
A
3FLWA_FLW
(MAPK14)
CMGC
Pamapimod
I
9
44
22
9
44
22
A
3FLQA_891
(MAPK14)
CMGC
FLS
I
8
25
20
8
25
20
A
3OCGA_OCG
(MAPK14)
CMGC
OCG
II
8
34
31
8
34
31
A
3FLSA_FLS
(MAPK14)
CMGC
FLS
I
8
26
20
8
26
20
A
3LHJA_LHJ
(MAPK14)
CMGC
LHJ
I
8
89
18
8
89
18
A
1W84A_L12
(MAPK14)
CMGC
3-(2-Pyridin...
I
6
10
25
6
10
25
A
3FMJA_FMJ
(MAPK14)
CMGC
Imidazo[1,2-...
I
6
5
36
6
5
36
A
3OC1A_BMU
(MAPK14)
CMGC
BMU
III
6
69
20
6
69
20
A
3GI3A_B10
(MAPK14)
CMGC
B10
II
6
8
20
6
8
20
A
3HVCA_GG5
(MAPK14)
CMGC
HMS3303H10
I
5
76
18
5
76
18
A
2ZB0A_GK3
(MAPK14)
CMGC
biphenyl ami...
II
5
43
21
5
43
21
A
3FSKA_RO6
(MAPK14)
CMGC
SU_14813
I
5
10
24
5
10
24
A
3GC7A_B45
(MAPK14)
CMGC
Sunitinib
I
5
63
16
5
63
16
A
3KF7A_L9G
(MAPK14)
CMGC
EDD
I
5
18
20
5
18
20
A
3BX5A_304
(MAPK14)
CMGC
BMS-640994
I
5
48
18
5
48
18
A
3FMNA_530
(MAPK14)
CMGC
Gefitinib
I
4
19
18
4
19
18
A
3HRBA_I39
(MAPK14)
CMGC
PTK_787
I
4
29
17
4
29
17
A
3HUBA_469
(MAPK14)
CMGC
Talmapimod
I
4
24
17
4
24
17
A
2BALA_PQA
(MAPK14)
CMGC
Ro-3201195
I
4
24
24
4
24
24
A
3HL7A_I47
(MAPK14)
CMGC
DB07943
I
4
17
21
4
17
21
A
3MPTA_1GK
(MAPK14)
CMGC
SMR000074150
I
4
7
22
4
7
22
A
1M7QA_DQO
(MAPK14)
CMGC
quinazolinon...
I
4
40
16
4
40
16
A
1WBWA_LI4
(MAPK14)
CMGC
LI4
I
4
4
32
4
4
32
A
1W7HA_3IP
(MAPK14)
CMGC
2-Amino-3-be...
I
3
3
32
3
3
32
A
3MW1A_MIH
(MAPK14)
CMGC
CAS745833_23_2
I
3
22
16
3
22
16
A
1OVEA_358
(MAPK14)
CMGC
Dihydro-quin...
I
3
26
16
3
26
16
A
3NWWA_3NW
(MAPK14)
CMGC
3NW
I
3
7
21
3
7
21
A
3FMMA_XI2
(MAPK14)
CMGC
XI2
I
2
15
12
2
15
12
A
1OUYA_094
(MAPK14)
CMGC
CAS745833_23_2
I
2
53
12
2
53
12
A
2GFSA_PQB
(MAPK14)
CMGC
aminopyrazol...
I
2
15
14
2
15
14
A
2I0HA_222
(MAPK14)
CMGC
MLN_8054
I
2
21
12
2
21
12
A
3FKNA_FKN
(MAPK14)
CMGC
XI2
I
2
5
12
2
5
12
A
3HLLA_I45
(MAPK14)
CMGC
PH-797804
I
2
63
12
2
63
12
A
3D7ZA_GK5
(MAPK14)
CMGC
DB07835
II
2
58
12
2
58
12
A
3FMLA_FML
(MAPK14)
CMGC
XI2
I
2
15
12
2
15
12
A
3FI4A_FI4
(MAPK14)
CMGC
SMR000463566
I
2
14
14
2
14
14
A
2ZAZA_GK1
(MAPK14)
CMGC
2zaz
I
1
2
12
1
2
12
A
3L8SA_BFF
(MAPK14)
CMGC
Kinome_3755
I
1
1
12
1
1
12
A
1ZZ2A_B11
(MAPK14)
CMGC
B11
I
1
3
12
1
3
12
A
3FL4A_FL4
(MAPK14)
CMGC
CGP79787 Ana...
I
1
6
12
1
6
12
A
3IW5A_DF3
(MAPK14)
CMGC
AC1NFSIE
I
1
1
12
1
1
12
A
2QD9A_LGF
(MAPK14)
CMGC
SU_14813
I
1
4
12
1
4
12
A
1WBOA_2CH
(MAPK14)
CMGC
2CH
I
1
1
12
1
1
12
E
22
3HV6A_R39
(MAPK14)
CMGC
R39
II
8
74
20
E
3HV6A_R39
(MAPK14)
CMGC
R39
II
8
74
20
8
74
20
E
1KV2A_B96
(MAPK14)
CMGC
Doramapimod
II
8
92
20
8
92
20
E
2BAKA_AQZ
(MAPK14)
CMGC
2bak
II
8
153
20
8
153
20
E
3HEGA_BAX
(MAPK14)
CMGC
Sorafenib
II
7
8
19
7
8
19
E
3HECA_STI
(MAPK14)
CMGC
Imatinib
II
7
158
20
7
158
20
E
3GCSA_BAX
(MAPK14)
CMGC
Sorafenib
II
7
8
19
7
8
19
E
3GCPA_SB2
(MAPK14)
CMGC
SB 203580
I
6
31
20
6
31
20
E
3HV3A_R49
(MAPK14)
CMGC
R49
II
5
39
20
5
39
20
E
3GCQA_1BU
(MAPK14)
CMGC
1BU
II
5
41
20
5
41
20
E
3O8TA_BMU
(MAPK14)
CMGC
BMU
III
4
66
17
4
66
17
E
3O8UA_BMU
(MAPK14)
CMGC
BMU
III
4
66
17
4
66
17
E
1KV1A_BMU
(MAPK14)
CMGC
BMU
III
4
66
17
4
66
17
E
3K3IA_JZJ
(MAPK14)
CMGC
Pyrazole-Bas...
II
4
12
15
4
12
15
E
2RG6A_287
(MAPK14)
CMGC
2rg6
II
4
159
15
4
159
15
E
2RG5A_279
(MAPK14)
CMGC
pyrrolo[2,1-...
II
3
107
14
3
107
14
E
3K3JA_F4C
(MAPK14)
CMGC
ABT_869
II
2
6
15
2
6
15
E
3LFBA_Z87
(MAPK14)
CMGC
diaryl urea ...
III
2
40
14
2
40
14
E
3CTQA_337
(MAPK14)
CMGC
acylated 2-a...
II
1
1
12
1
1
12
E
3LFEA_Z84
(MAPK14)
CMGC
diaryl urea ...
II
1
5
12
1
5
12
E
3LFDA_Z85
(MAPK14)
CMGC
diaryl urea ...
III
1
5
12
1
5
12
E
3IW8A_HIZ
(MAPK14)
CMGC
thieno[3,2-d...
II
1
2
12
1
2
12
E
3LFCA_Z86
(MAPK14)
CMGC
diaryl urea ...
III
1
5
12
1
5
12
F
22
3HV4A_L51
(MAPK14)
CMGC
L51
II
2
37
15
F
3HV4A_L51
(MAPK14)
CMGC
L51
II
2
37
15
2
37
15
F
3HV5A_R24
(MAPK14)
CMGC
R24
II
2
28
15
2
28
15
F
1W82A_L10
(MAPK14)
CMGC
AC1LCVRE
II
2
56
15
2
56
15
F
3E93A_19B
(MAPK14)
CMGC
AMG_706
II
2
42
15
2
42
15
F
3KQ7A_KQ7
(MAPK14)
CMGC
BIRB_796
II
2
87
15
2
87
15
F
3GCVA_SS6
(MAPK14)
CMGC
quinazoline-...
II
2
38
15
2
38
15
F
3GCUA_R48
(MAPK14)
CMGC
L51
II
2
38
15
2
38
15
F
3BV3A_P39
(MAPK14)
CMGC
BIRB_796
II
2
138
15
2
138
15
F
1W83A_L11
(MAPK14)
CMGC
AC1LCVRH
II
1
2
12
1
2
12
F
3NNUA_EDB
(MAPK14)
CMGC
EDD
II
1
11
12
1
11
12
F
3NNVA_437
(MAPK14)
CMGC
diaryl urea ...
II
1
2
12
1
2
12
F
3NNWA_EDD
(MAPK14)
CMGC
EDD
II
1
36
12
1
36
12
F
3NNXA_EDD
(MAPK14)
CMGC
EDD
II
1
36
12
1
36
12
F
3D83A_GK6
(MAPK14)
CMGC
3d83
II
1
62
12
1
62
12
F
1WBTA_WBT
(MAPK14)
CMGC
WBT
II
1
8
12
1
8
12
F
1WBSA_LI2
(MAPK14)
CMGC
LI2
II
1
8
12
1
8
12
F
3HP2A_P36
(MAPK14)
CMGC
1-benzyl-4-(...
I
1
30
12
1
30
12
F
1WBNA_L09
(MAPK14)
CMGC
L09
II
1
5
12
1
5
12
F
1WBVA_LI3
(MAPK14)
CMGC
LI3
III
1
5
12
1
5
12
F
2BAJA_1PP
(MAPK14)
CMGC
2-((1 R-isop...
II
1
1
12
1
1
12
F
2BAQA_PQB
(MAPK14)
CMGC
aminopyrazol...
I
1
15
12
1
15
12
F
3IW6A_PP0
(MAPK14)
CMGC
MLS000097106
I
1
1
12
1
1
12