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Diseases
Inhibitor-Anchor Map
Family Anchors
Kinase-Inhibitor Family
Template
Protein
Surface
Ribbon
Inhibitor
ATP Location
Pocket
ATP
NLP
HAP
CLP
SP
Summary of query kinase
Query kinase
GSK3A (
P49840
)
Kinase group
CMGC
Number of conformation types
0
Number of structural templates
110 (
Total 331 inhibitors
)
Select
Template
Comformation
Type
No. of
Templates
Representative
Template
Kinase
Group
Representative
Inhibitor
Inhibitor
Type
No. of
Kinases
No. of
Inhibitors
No. of
Diseases
A
62
2OW3A_BIM
(GSK3B)
CMGC
LY_333531
I
62
139
51
A
2OW3A_BIM
(GSK3B)
CMGC
LY_333531
I
62
139
51
62
139
51
A
3IW4A_LW4
(PRKCA)
CMGC
Sotrastaurin
I
52
119
49
52
119
49
A
1Q4LA_679
(GSK3B)
CMGC
I-5
I
3
26
7
3
26
7
A
1VYWA_292
(CDK2)
CMGC
PNU-292137 I...
I
20
91
38
20
91
38
A
1AQ1A_STU
(CDK2)
CMGC
staurosporine
I
195
76
118
195
76
118
A
1XJDA_STU
(PRKCQ)
CMGC
staurosporine
I
121
101
106
121
101
106
A
1NVRA_STU
(CHEK1)
CMGC
staurosporine
I
179
71
79
179
71
79
A
1NXKA_STU
(MAPKAPK2)
CMGC
staurosporine
I
110
67
51
110
67
51
A
3L8XA_N4D
(MAPK14)
CMGC
3cg2
I
91
104
65
91
104
65
A
1Q3DA_STU
(GSK3B)
CMGC
staurosporine
I
115
71
61
115
71
61
A
1YVJA_4ST
(JAK3)
CMGC
staurosporine
I
96
90
126
96
90
126
A
1NVQA_UCN
(CHEK1)
CMGC
UCN 02
I
179
65
79
179
65
79
A
1PKDA_UCN
(CDK2)
CMGC
UCN 02
I
195
67
118
195
67
118
A
2JBPA_P4O
(MAPKAPK2)
CMGC
2jbo
I
18
130
30
18
130
30
A
3R2YA_P4O
(MAPKAPK2)
CMGC
2jbo
I
18
130
30
18
130
30
A
2JBOA_P4O
(MAPKAPK2)
CMGC
2jbo
I
18
130
30
18
130
30
A
2V7OA_DRN
(CAMK2G)
CMGC
bisindolylma...
I
23
51
16
23
51
16
A
2HY81_1ST
(PAK1)
CMGC
UCN 02
I
58
20
75
58
20
75
A
3MVLA_38P
(MAPK14)
CMGC
38P
I
50
308
44
50
308
44
A
3NLBA_5BE
(CHEK1)
CMGC
38P
I
45
115
49
45
115
49
A
3M2WA_L8I
(MAPKAPK2)
CMGC
Sunitinib
I
84
90
47
84
90
47
A
2J51A_DKI
(SLK)
CMGC
5-AMINO-3-{[...
I
90
11
103
90
11
103
A
2JFLA_DKI
(SLK)
CMGC
5-AMINO-3-{[...
I
90
11
103
90
11
103
A
2WIHA_P48
(CDK2)
CMGC
VX_680
I
111
425
105
111
425
105
A
2WU6A_DKI
(CLK3)
CMGC
5-AMINO-3-{[...
I
26
9
26
26
9
26
A
3DS6A_A17
(MAPK14)
CMGC
3ds6
II
21
146
34
21
146
34
A
3L1SA_Z92
(GSK3B)
CMGC
AN-988/42110...
I
5
33
9
5
33
9
A
3BLRA_CPB
(CDK9)
CMGC
BIIVYFLTOXDA...
I
48
17
41
48
17
41
A
2R3NA_SCZ
(CDK2)
CMGC
AC1LZZHM
I
46
175
57
46
175
57
A
3EQFA_KSA
(MAP2K1)
CMGC
k-252a
I
42
51
57
42
51
57
A
2VTNA_LZ7
(CDK2)
CMGC
pyrazole ami...
I
8
48
24
8
48
24
A
1Q3WA_ATU
(GSK3B)
CMGC
alsterpaullone
I
24
28
19
24
28
19
A
3ITZA_P66
(MAPK14)
CMGC
P66
II
15
102
25
15
102
25
A
1R0EA_DFN
(GSK3B)
CMGC
HMS3401D14
I
17
17
17
17
17
17
A
2B55A_D31
(CDK2)
CMGC
D31
I
27
87
53
27
87
53
A
3MVMA_39P
(MAPK14)
CMGC
39P
I
24
247
38
24
247
38
A
3EJ1A_5BP
(CDK2)
CMGC
AC1OCFRV
I
46
92
62
46
92
62
A
1GIHA_1PU
(CDK2)
CMGC
1PU
I
13
60
35
13
60
35
A
2VU3A_LZE
(CDK2)
CMGC
AT7519
I
35
22
29
35
22
29
A
3D0EA_G93
(AKT2)
CMGC
9-N-ethyl-8-...
I
30
15
45
30
15
45
A
3NR9A_NR9
(CLK2)
CMGC
Cdk1 Inhibit...
I
6
5
19
6
5
19
A
2XIKA_J60
(STK25)
CMGC
SU11652
I
59
49
65
59
49
65
A
2JDRA_L20
(AKT2)
CMGC
A-443654
I
44
255
61
44
255
61
A
1Q5KA_TMU
(GSK3B)
CMGC
AR-A014418
I
2
4
6
2
4
6
A
2ZB1A_GK4
(MAPK14)
CMGC
biphenyl ami...
II
55
57
54
55
57
54
A
2E9VA_85A
(CHEK1)
CMGC
macrocyclic ...
I
14
121
27
14
121
27
A
3GFEA_P37
(MAPK14)
CMGC
DB08349
I
11
83
29
11
83
29
A
3E92A_G6A
(MAPK14)
CMGC
3e92
I
56
59
55
56
59
55
A
3HA8A_5JZ
(MAPK14)
CMGC
DEL-B, 14b
I
59
89
62
59
89
62
A
3LHJA_LHJ
(MAPK14)
CMGC
LHJ
I
8
89
18
8
89
18
A
3IPHA_G11
(MAPK14)
CMGC
HMS3303K05
I
57
108
55
57
108
55
A
1ZYSA_199
(CHEK1)
CMGC
2,4-Diamino-...
I
31
92
52
31
92
52
A
2JEDA_LG8
(PRKCQ)
CMGC
5-Arylidene-...
I
67
19
87
67
19
87
A
1UV5A_BRW
(GSK3B)
CMGC
6-bromoindir...
I
27
37
28
27
37
28
A
1OUKA_084
(MAPK14)
CMGC
1ouk
I
24
139
46
24
139
46
A
2OWBA_626
(PLK1)
CMGC
2j4z
I
10
48
22
10
48
22
A
2BHEA_BRY
(CDK2)
CMGC
BRY
I
51
31
35
51
31
35
A
3KGAA_LX9
(MAPKAPK2)
CMGC
LX9
I
14
42
21
14
42
21
A
2VTQA_LZA
(CDK2)
CMGC
pyrazole dia...
I
36
25
31
36
25
31
A
1NVSA_UCM
(CHEK1)
CMGC
SB218078
I
97
6
53
97
6
53
A
3KVWA_IRB
(DYRK2)
CMGC
CI_1040
I
15
36
12
15
36
12
A
2VTTA_LZD
(CDK2)
CMGC
pyrazole dia...
I
158
42
111
158
42
111
B
48
3LFSA_A07
(CDK2)
CMGC
DNC010588
I
14
111
31
B
3LFSA_A07
(CDK2)
CMGC
DNC010588
I
14
111
31
14
111
31
B
3LAUA_OFI
(AURKA)
CMGC
DNC010577
I
12
112
35
12
112
35
B
3LFNA_A27
(CDK2)
CMGC
DNC010577
I
14
98
33
14
98
33
B
3LFQA_A28
(CDK2)
CMGC
DNC010588
I
10
99
30
10
99
30
B
1UU8A_BI1
(PDPK1)
CMGC
bisindolylma...
I
83
189
65
83
189
65
B
1ZRZA_BI1
(PRKCI)
CMGC
bisindolylma...
I
52
150
47
52
150
47
B
3ORZA_BI4
(PDPK1)
CMGC
bisindolylma...
I
82
178
65
82
178
65
B
3OTUA_BI4
(PDPK1)
CMGC
bisindolylma...
I
82
178
65
82
178
65
B
1UU7A_BI2
(PDPK1)
CMGC
bisindolylma...
I
82
178
65
82
178
65
B
1UVRA_BI8
(PDPK1)
CMGC
Ro 31-7549
I
82
181
65
82
181
65
B
1UU9A_BI3
(PDPK1)
CMGC
3-[1-(3-AMIN...
I
83
180
69
83
180
69
B
2OJGA_19A
(MAPK1)
CMGC
Oprea1_828620
I
8
75
28
8
75
28
B
1OIQA_HDU
(CDK2)
CMGC
AC1L9L2U
I
14
56
31
14
56
31
B
3COHA_83H
(AURKA)
CMGC
AKI-001
I
79
88
65
79
88
65
B
1UU3A_LY4
(PDPK1)
CMGC
Ruboxistaurin
I
71
117
57
71
117
57
B
1OKYA_STU
(PDPK1)
CMGC
staurosporine
I
179
67
109
179
67
109
B
1OKZA_UCN
(PDPK1)
CMGC
UCN 02
I
179
60
109
179
60
109
B
3GOKA_P4O
(MAPKAPK2)
CMGC
2jbo
I
20
134
35
20
134
35
B
3IO7A_1P5
(JAK2)
CMGC
CP_690550
I
24
65
60
24
65
60
B
2P3GX_F10
(MAPKAPK2)
CMGC
Pyrrolopyrid...
I
8
89
10
8
89
10
B
2W1FA_L0F
(AURKA)
CMGC
DB08066
I
17
40
35
17
40
35
B
2W1HA_L0H
(CDK2)
CMGC
DB08066
I
20
43
42
20
43
42
B
3CGOA_JNO
(MAPK10)
CMGC
DB08026
I
13
32
21
13
32
21
B
3E63A_5B2
(JAK2)
CMGC
5-phenyl-1H-...
I
15
29
39
15
29
39
B
3FUPA_MI1
(JAK2)
CMGC
CP690550
I
16
27
32
16
27
32
B
3AMAA_SKE
(PRKACA)
CMGC
JNJ-7706621
I
46
26
35
46
26
35
B
1TVOA_FRZ
(MAPK1)
CMGC
FR-180204
I
9
17
23
9
17
23
B
2XCKA_MH4
(PDPK1)
CMGC
MH4
I
46
431
75
46
431
75
B
3NRMA_NRM
(AURKA)
CMGC
CAS404828_08_6
I
32
33
60
32
33
60
B
3QD0A_3Q4
(PDPK1)
CMGC
(3s,6r)-1-[2...
I
28
114
63
28
114
63
B
3P9JA_P9J
(AURKA)
CMGC
4-[(5-Methyl...
I
32
50
54
32
50
54
B
1GIIA_1PU
(CDK2)
CMGC
1PU
I
12
60
29
12
60
29
B
3L9MA_L9M
(PRKACA)
CMGC
VX_680
I
37
65
42
37
65
42
B
3MTLA_FEF
(PCTK1)
CMGC
indirubin de...
I
16
3
23
16
3
23
B
2R3KA_SCQ
(CDK2)
CMGC
2r3j
I
28
95
49
28
95
49
B
3L9NA_L9N
(PRKACA)
CMGC
A_674563
I
10
63
36
10
63
36
B
2E14A_FRR
(MAPK1)
CMGC
L-783279
I
6
6
21
6
6
21
B
1PF8A_SU9
(CDK2)
CMGC
SU 9516
I
25
19
33
25
19
33
B
2BMCA_MPY
(AURKA)
CMGC
PHA-680632
I
107
108
107
107
108
107
B
3PY0A_SU9
(CDK2)
CMGC
SU 9516
I
25
19
33
25
19
33
B
3PY1A_SU9
(CDK2)
CMGC
SU 9516
I
25
19
33
25
19
33
B
2J4ZA_626
(AURKA)
CMGC
2j4z
I
13
51
25
13
51
25
B
2FVDA_LIA
(CDK2)
CMGC
[4-Amino-2-[...
I
39
16
29
39
16
29
B
3EFWA_AK8
(AURKA)
CMGC
3efw
I
100
59
105
100
59
105
B
2PE2A_464
(PDPK1)
CMGC
Indolinone b...
I
134
156
104
134
156
104
B
2XRUA_400
(AURKA)
CMGC
VX_680
I
33
152
63
33
152
63
B
2R3JA_SCJ
(CDK2)
CMGC
2r3j
I
27
99
49
27
99
49
B
2PE0A_39Z
(PDPK1)
CMGC
2pe0
I
20
2
27
20
2
27